发明申请
US20060166824A1 Avermectin and avemectin monosaccharide derivatives substituted in the 4"-or 4'-position having pesticidal properties
有权
在4“ - 或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物
- 专利标题: Avermectin and avemectin monosaccharide derivatives substituted in the 4"-or 4'-position having pesticidal properties
- 专利标题(中): 在4“ - 或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物
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申请号: US10543638申请日: 2004-01-30
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公开(公告)号: US20060166824A1公开(公告)日: 2006-07-27
- 发明人: Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Pierre Jung
- 申请人: Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Pierre Jung
- 优先权: GB0302310.8 20030131
- 国际申请: PCT/EP04/00900 WO 20040130
- 主分类号: A01N43/04
- IPC分类号: A01N43/04 ; A61K31/7048
摘要:
Disclosed are compounds of the formula in which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —S02—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2 is R3-Z-, R3—O-Z-, R4 or -Z-N(R6)(R7); Q is O or —N—R5; R3 and R4 are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6 and R7 are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.
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