中科微点-全球专利检索

  1. Login
  2. Sign Up

Search Results

47 records (took 0.028 seconds)

    Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position
    3.
    发明授权
    Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position 有权
    在4“ - 或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物

    公开(公告)号：US08017589B2

    公开(公告)日：2011-09-13

    申请号：US12768280

    申请日：2010-04-27

    Applicant: Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Franz Hueter ,  Pierre Jung

    Inventor： Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Franz Hueter ,  Pierre Jung

    IPC: A61K31/70 ,  C07H17/04

    CPC classification number: C07H17/08 ,  A61K31/7042

    Abstract: What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.

    Abstract translation: 描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基， 卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基， 芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或 盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

    "> AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4
    4.
    发明申请
    AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4"-OR 4'-POSITION 有权
    在4“-OR 4'-位置具有烷氧基取代基的AVERMECTIN B1和AVERMECTIN B1单糖衍生物

    公开(公告)号：US20100210574A1

    公开(公告)日：2010-08-19

    申请号：US12768280

    申请日：2010-04-27

    Applicant: Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Franz Hueter ,  Pierre Jung

    Inventor： Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Franz Hueter ,  Pierre Jung

    IPC: A01N43/16 ,  C07H17/08 ,  A01P17/00

    CPC classification number: C07H17/08 ,  A61K31/7042

    Abstract: What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.

    Abstract translation: 描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基， 卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基， 芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或 盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

    Avermectin and avemectin monosaccharide derivatives substituted in the 4″- or 4′-position having pesticidal properties
    5.
    发明授权
    Avermectin and avemectin monosaccharide derivatives substituted in the 4″- or 4′-position having pesticidal properties 有权
    在4“或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物

    公开(公告)号：US07632820B2

    公开(公告)日：2009-12-15

    申请号：US10543638

    申请日：2004-01-30

    Applicant: Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

    Inventor： Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

    IPC: A01N43/04 ,  A61K31/40 ,  A61K31/335 ,  A61K31/70 ,  A61K31/397 ,  A61K31/445 ,  A61K31/44 ,  A01N43/38

    CPC classification number: A01N43/90 ,  C07H17/08

    Abstract: Disclosed are compounds of the formulain which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —SO2—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2 is R3-Z-, R3—O-Z-, R4 or -Z-N(R6)(R7); Q is O or —N—R5; R3 and R4 are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6 and R7 are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.

    Abstract translation: 公开了n为0或1的甲醛化合物; X-Y是-CH-CH-或-CH 2 -CH 2 - ; Z是-C（-O） - ， - C（-S） - 或-SO 2 - ; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; R2为R3-Z-，R3-O-Z-，R4或-Z-N（R6）（R7）; Q是O或-N-R5; R 3和R 4例如是H，C 1 -C 12烷基，C 2 -C 12烯基，C 2 -C 12炔基，C 3 -C 12环烷基，C 5 -C 12环烯基，芳基或杂环基; R5是例如H，C1-C8烷基，羟基-C1-C8烷基，C3-C8环烷基，C2-C8链烯基，C2-C8炔基，苯基或苄基; R 6和R 7为例如未取代的或未被取代的一价或五价取代的C 1 -C 12烷基，未被取代的或一至五取代的C 2 -C 12链烯基或（如果合适的话）E / Z异构体，E / Z异构体混合物和/或其互变异构体， 在每种情况下以游离形式或盐形式，都可用作农药。

    "> Avermectin and avemectin monosaccharide derivatives substituted in the 4
    6.
    发明申请
    Avermectin and avemectin monosaccharide derivatives substituted in the 4"-or 4'-position having pesticidal properties 有权
    在4“ - 或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物

    公开(公告)号：US20060166824A1

    公开(公告)日：2006-07-27

    申请号：US10543638

    申请日：2004-01-30

    Applicant: Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

    Inventor： Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

    IPC: A01N43/04 ,  A61K31/7048

    CPC classification number: A01N43/90 ,  C07H17/08

    Abstract: Disclosed are compounds of the formula in which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —S02—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2 is R3-Z-, R3—O-Z-, R4 or -Z-N(R6)(R7); Q is O or —N—R5; R3 and R4 are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6 and R7 are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.

    Abstract translation: 公开了下式的化合物，其中n为0或1; X-Y是-CH-CH-或-CH 2 -CH 2 - 。 Z是-C（-O） - ， - C（-S） - 或-SO 2 - 。 R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 1 -C 12烷基，C 3 -C 12烷基， 环烷基或C 2 -C 12 - 烯基; 和R 2是R 3 -Z-，R 3 -OZ-，R 4或-ZN（ R 6）（R 7）; Q是O或-N-R 5; R 3和R 4是例如H，C 1 -C 12烷基，C 2， C 1 -C 12亚烷基，C 2 -C 12炔基，C 3 -C 12链烯基，C 2 -C 12亚炔基，C 3 -C 12亚烷基， 12个环烷基，C 5 -C 12环烯基，芳基或杂环基; R 5是例如H，C 1 -C 8烷基，羟基-C 1 -C 3 C 1 -C 8烷基，C 3 -C 8环烷基，C 2 -C 8链烯基，C 1 -C 8烷基， C 2 -C 8炔基，苯基或苄基; R 6和R 7是例如H，未取代的或一至五取代的C 1 -C 12 - 烷基，未取代的或一至五取代的C 2 -C 12链烯基，或者如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体， 在每种情况下以游离形式或盐形式，都可用作农药。

    "> Avermectin b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substitutent in the 4
    7.
    发明申请
    Avermectin b1 and avermectin b1 monosaccharide derivatives having an alkoxymethyl substitutent in the 4"-or 4'-position 有权

    公开(公告)号：US20060148729A1

    公开(公告)日：2006-07-06

    申请号：US10539274

    申请日：2003-12-19

    Applicant: Peter Maienfisch ,  Fiona Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Hueter ,  Pierre Jung

    Inventor： Peter Maienfisch ,  Fiona Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Hueter ,  Pierre Jung

    IPC: A01N43/04 ,  C07H17/08

    CPC classification number: C07H17/08 ,  A61K31/7042

    Abstract: What is described are a compound of the formula (I): wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —N02, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12 alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)-Z-R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.

    Microbiocidal heterocycles
    9.
    发明授权
    Microbiocidal heterocycles 有权
    微生物杂环

    公开(公告)号：US08367844B2

    公开(公告)日：2013-02-05

    申请号：US13390023

    申请日：2010-08-06

    Applicant: Sarah Sulzer-Mosse ,  Clemens Lamberth ,  Laura Quaranta ,  Mathias Stephan Respondek

    Inventor： Sarah Sulzer-Mosse ,  Clemens Lamberth ,  Laura Quaranta ,  Mathias Stephan Respondek

    IPC: A01N43/40 ,  A01N43/36 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  C07D401/02 ,  C07D401/14 ,  C07D403/02 ,  C07D403/14 ,  C07D207/04 ,  C07D231/10 ,  C07D241/04

    CPC classification number: C07D401/14 ,  C07D231/12 ,  C07D401/04 ,  C07D401/06 ,  C07D401/12

    Abstract: The present invention relates to heterocyclic compounds of formula I which have microbiocidal activity, in particular fungicidal activity as well as methods of using the compounds of formula (I) to control microbes: wherein A is x-C(R10R11)—C(═O)—, x-C(R12R13)—C(═S)—, x-O—C(═O)—, x-O—C(═S)—, x-N(R14)—C(═O)—, x-N(R15)—C(═S)—, x-C(R16R17)—SO2— or X—N═C(R30)—, in each case x indicates the bond that is connected to R1; T is CR18 or N; Y1, Y2, Y3, and Y4 are independently CR19 or N; Q is O or S; n is 1 or 2; p is 1 or 2, providing that when n is 2, p is 1. R1 is phenyl, pyridyl, imidazolyl, or pyrazolyl; wherein the phenyl, pyridyl, imidazolyl and pyrazolyl are each optionally substituted by 1 to 3 substituents independently selected from C1-C4 alkyl, C1-C4 haloalkyl, halogen, cyano, hydroxy and amino; R2, R3, R4, R5, R6, R7, R10, R11, R12, R13, R16, R17, R18, R19 and R30 each independently are hydrogen, halogen, cyano, C1-C4alkyl, or C1-C4haloalkyl; R8, R14 and R15 each independently are hydrogen or C1-C4alkyl; and R9 is phenyl, benzyl or group (a): wherein the phenyl, benzyl and group (a) are each optionally substituted with 1 to 3 substituents independently selected from C1-C4 alkyl, C1-C4 haloalkyl, halogen, cyano, hydroxy and amino; or a salt or a N-oxide thereof.

    Abstract translation: 本发明涉及具有杀微生物活性，特别是杀真菌活性的式I的杂环化合物以及使用式（I）化合物来控制微生物的方法：其中A是xC（R10R11）-C（= O） - ，xC（R12R13）-C（= S） - ，xO-C（= O） - ，xO-C（= S） - ，xN（R14）-C（= O） - ，xN（R15）-C （X）（R 16 R 17）-SO 2 - 或X-N = C（R 30） - ，在各种情况下，x表示与R1连接的键; T为CR18或N; Y1，Y2，Y3和Y4独立地为CR19或N; Q是O或S; n为1或2; p为1或2，条件是当n为2时，p为1. R1为苯基，吡啶基，咪唑基或吡唑基; 其中苯基，吡啶基，咪唑基和吡唑基各自任选被1至3个独立地选自C 1 -C 4烷基，C 1 -C 4卤代烷基，卤素，氰基，羟基和氨基的取代基取代; R2，R3，R4，R5，R6，R7，R10，R11，R12，R13，R16，R17，R18，R19和R30各自独立地为氢，卤素，氰基，C1-C4烷基或C1-C4卤代烷基; R8，R14和R15各自独立地为氢或C1-C4烷基; 并且R 9为苯基，苄基或基团（a）：其中苯基，苄基和基团（a）各自任选被1至3个独立地选自C 1 -C 4烷基，C 1 -C 4卤代烷基，卤素，氰基，羟基和 氨基; 或其盐或N-氧化物。

Patent Agency Ranking