Invention Application
US20080021017A1 2-Phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
有权
2-苯基-1- [4-(2-氨基乙氧基) - 苄基] - 吲哚作为雌激素剂
- Patent Title: 2-Phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
- Patent Title (中): 2-苯基-1- [4-(2-氨基乙氧基) - 苄基] - 吲哚作为雌激素剂
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Application No.: US11820735Application Date: 2007-06-20
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Publication No.: US20080021017A1Publication Date: 2008-01-24
- Inventor: Chris Miller , Michael Collini , Bach Tran , Arthur Santilli
- Applicant: Chris Miller , Michael Collini , Bach Tran , Arthur Santilli
- Applicant Address: US NJ Madison
- Assignee: Wyeth
- Current Assignee: Wyeth
- Current Assignee Address: US NJ Madison
- Main IPC: A61K31/404
- IPC: A61K31/404 ; A61K31/4523 ; A61K31/496 ; A61K31/55 ; A61P15/00 ; A61P17/10 ; A61P19/10 ; A61P25/28 ; A61P35/00 ; A61P9/00
![2-Phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents](/abs-image/US/2008/01/24/US20080021017A1/abs.jpg.150x150.jpg)
Abstract:
The present invention relates to new 2-Phenyl-1-[4-(2-Aminoethoxy)-Benzyl]-Indole compounds having the general structures below: which are useful in contraception and in treating melanoma, osteoporosis, acne, dysfunctional uterine bleeding, endometrial polyps, benign breast disease, adenomyosis, infertility, endometriosis, endometrial cancer, polycystic ovary syndrome, cardiovascular disease, Alzheimer's disease, cognitive decline, central nervous system disorders, central nervous system cancers, leukemia, endometrial ablations, chronic renal disease, chronic hepatic disease, coagulation diseases and disorders, hypocalcemia, hypercalcemia, Paget's disease, osteomalacia, osteohalisteresis, and multiple myeloma.
Public/Granted literature
- US07449455B2 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents Public/Granted day:2008-11-11
Information query
IPC分类: