发明申请
- 专利标题： SNAR PROCESS FOR PREPARING BENZIMIDAZOLE COMPOUNDS
- 专利标题（中）： 制备苯并咪唑化合物的SNAR方法
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申请号： US11917998申请日： 2006-06-21
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公开(公告)号： US20100130748A1公开(公告)日： 2010-05-27
- 发明人: John Demattei , Sagar Shakya , Paul J. Nichols , Bradley R. Barnett , Bruno P. Hache , Matthew Charles Evans , James Gair Ford , John Leonard
- 申请人： John Demattei , Sagar Shakya , Paul J. Nichols , Bradley R. Barnett , Bruno P. Hache , Matthew Charles Evans , James Gair Ford , John Leonard
- 申请人地址： US CO Boulder SE Sodertalje
- 专利权人： ARRAY BIOPHARMA INC.,ASTRAZENECA AB
- 当前专利权人： ARRAY BIOPHARMA INC.,ASTRAZENECA AB
- 当前专利权人地址： US CO Boulder SE Sodertalje
- 国际申请： PCT/US2006/023986 WO 20060621
- 主分类号： C07D235/04
- IPC分类号： C07D235/04
摘要：
Provided are methods for the synthesis of heterocyclic compounds such as benzimidazole carboxylic acid core structures having Formula Ia-2 and their synthetic intermediates: wherein X1, X2, X5, R1, R2 and R4 are as defined herein. Compounds of Formula Ia-2 and their synthetic intermediates can be used to prepare heterocyclic derivatives such as benzimidazole derivatives.
公开/授权文献
- US08183385B2 SNAR process for preparing benzimidazole compounds 公开/授权日：2012-05-22
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