发明申请
US20100249187A1 NOVEL DICARBOXYLIC ACID DERIVATIVES AS S1P1 RECEPTOR AGONISTS
有权
新型二羧酸衍生物作为S1P1受体激动剂
- 专利标题： NOVEL DICARBOXYLIC ACID DERIVATIVES AS S1P1 RECEPTOR AGONISTS
- 专利标题（中）： 新型二羧酸衍生物作为S1P1受体激动剂
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申请号： US12664718申请日： 2008-06-16
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公开(公告)号： US20100249187A1公开(公告)日： 2010-09-30
- 发明人: Marc Capet , Nicolas Levoin , Isabelle Berrebi-Bertrand , Philippe Robert , Jean-Charles Schwartz , Jeanne-Marie Lecomte , Jayraj Dilipbhal Aradhye , Muthukumaran Natarajan Pillai , Bhavesh Mohanbhai Panchal , Jignesh Kantilal Jivani , Biswajit Samanta , Ranjan Kumar Pal , Rajamannar Thennati
- 申请人： Marc Capet , Nicolas Levoin , Isabelle Berrebi-Bertrand , Philippe Robert , Jean-Charles Schwartz , Jeanne-Marie Lecomte , Jayraj Dilipbhal Aradhye , Muthukumaran Natarajan Pillai , Bhavesh Mohanbhai Panchal , Jignesh Kantilal Jivani , Biswajit Samanta , Ranjan Kumar Pal , Rajamannar Thennati
- 优先权： EP07290748.8 20070615
- 国际申请： PCT/EP2008/057571 WO 20080616
- 主分类号： A61K31/4545
- IPC分类号： A61K31/4545 ; C07D401/14 ; C07D213/02 ; A61K31/454 ; A61P37/06
摘要：
The present invention relates to new compounds of formula (I) possessing agonistic activity at sphingosine-1-phosphate (S1P) receptors, their process of preparation and their use as immunosuppressive agents. The invention is also directed to pharmaceutical compositions containing these compounds and use of these compounds for treatment/prevention of immune mediated diseases and conditions or inflammatory diseases and conditions.
公开/授权文献
- US08809539B2 Dicarboxylic acid derivatives as S1P1 receptor agonists 公开/授权日：2014-08-19