发明申请
US20100317645A1 SUBSTITUTED DIAZEPINE SULFONAMIDES AS BOMBESIN RECEPTOR SUBTYPE-1 MODULATORS
有权
替代亚硫酸荧光素作为BOMBESIN受体亚型1调节剂
- 专利标题： SUBSTITUTED DIAZEPINE SULFONAMIDES AS BOMBESIN RECEPTOR SUBTYPE-1 MODULATORS
- 专利标题（中）： 替代亚硫酸荧光素作为BOMBESIN受体亚型1调节剂
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申请号： US12517836申请日： 2007-12-07
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公开(公告)号： US20100317645A1公开(公告)日： 2010-12-16
- 发明人: Robert K. Baker , Linda L. Chang , Marc Chioda , Harry R. Chobanian , Ying-Duo Gao , Yan Guo , Linus S. Lin , Ping Liu , Ravi P. Nargund , Kathleen M. Rupprecht , Shouwu Miao
- 申请人： Robert K. Baker , Linda L. Chang , Marc Chioda , Harry R. Chobanian , Ying-Duo Gao , Yan Guo , Linus S. Lin , Ping Liu , Ravi P. Nargund , Kathleen M. Rupprecht , Shouwu Miao
- 国际申请： PCT/US2007/025104 WO 20071207
- 主分类号： A61K31/551
- IPC分类号： A61K31/551 ; C07D487/04 ; C07D498/14 ; C07D487/14 ; A61P3/10 ; A61P3/04
摘要：
Certain novel substituted diazepine sulfonamides are ligands of the human bombesin receptor and, in particular, are selective ligands of the human bombesin receptor subtype-3 (BRS-3). They are therefore useful for the treatment, control, or prevention of diseases and disorders responsive to the modulation of BRS-3, such as obesity, and diabetes.
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