发明申请
- 专利标题: PHENYLPYRAZOLE DERIVATIVES
- 专利标题(中): 苯并噻唑衍生物
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申请号: US12951978申请日: 2010-11-22
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公开(公告)号: US20110065668A1公开(公告)日: 2011-03-17
- 发明人: Toshio NAKAMURA , Makoto Tatsuzuki , Dai Nozawa , Tomoko Tamita , Seiji Masuda , Hiroshi Ohta , Shuhei Kashiwa , Aya Fujino , Shigeyuki Chaki , Toshiharu Shimazaki
- 申请人: Toshio NAKAMURA , Makoto Tatsuzuki , Dai Nozawa , Tomoko Tamita , Seiji Masuda , Hiroshi Ohta , Shuhei Kashiwa , Aya Fujino , Shigeyuki Chaki , Toshiharu Shimazaki
- 申请人地址: JP Tokyo
- 专利权人: TAISHO PHARMACEUTICAL CO., LTD.
- 当前专利权人: TAISHO PHARMACEUTICAL CO., LTD.
- 当前专利权人地址: JP Tokyo
- 优先权: JP2007294040 20071113; JP2008153736 20080612
- 主分类号: A61K31/695
- IPC分类号: A61K31/695 ; A61K31/415 ; A61K31/5377 ; A61K31/553 ; A61P25/28 ; A61P25/18 ; A61P3/10 ; A61P25/24 ; A61P25/08 ; A61P25/00
摘要:
The present invention provides a prophylactic or therapeutic agent for dementia, Alzheimer's disease, attention-deficit hyperactivity disorder, schizophrenia, eating disorders, obesity, diabetes, hyperlipidemia, sleep disorders, narcolepsy, sleep apnea syndrome, circadian rhythm disorder, depression, allergic rhinitis or other diseases.A phenylpyrazole derivative represented by formula (1) or a pharmaceutically acceptable salt thereof: {wherein R1 and R2, which may be the same or different, each represent C1-C6 alkyl or C3-C8 cycloalkyl, or R1 and R2 are attached to each other together with their adjacent nitrogen atom to form a 4- to 7-membered saturated heterocyclic ring (wherein said saturated heterocyclic ring may be substituted with halogen or C1-C6 alkyl), n represents an integer of 0 to 2, T represents a hydrogen atom, halogen or C1-C6 alkyl, and R represents formula (I): or the like}.
公开/授权文献
- US08193176B2 Phenylpyrazole derivatives 公开/授权日:2012-06-05
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