发明申请
- 专利标题： TRIAZOLOPYRIDINE DERIVATIVES
- 专利标题（中）： 三唑吡啶衍生物
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申请号： US13512721申请日： 2010-11-26
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公开(公告)号： US20130121994A1公开(公告)日： 2013-05-16
- 发明人: Marcus Koppitz , Volker Schulze , Dirk Kosemund , Hartmut Schirok , Benjamin Bader , Philip Lienau , Tobias Marquardt , Christof Wegscheid-Gerlach , Gerhard Siemeister , Stefan Prechtl , Antje Margret Wengner , Ulf Bömer
- 申请人： Marcus Koppitz , Volker Schulze , Dirk Kosemund , Hartmut Schirok , Benjamin Bader , Philip Lienau , Tobias Marquardt , Christof Wegscheid-Gerlach , Gerhard Siemeister , Stefan Prechtl , Antje Margret Wengner , Ulf Bömer
- 申请人地址： DE Monheim
- 专利权人： BAYER INTELLECTUAL PROPERTY GMBH
- 当前专利权人： BAYER INTELLECTUAL PROPERTY GMBH
- 当前专利权人地址： DE Monheim
- 优先权： EP09075534.9 20091130
- 国际申请： PCT/EP10/68298 WO 20101126
- 主分类号： C07D471/04
- IPC分类号： C07D471/04 ; A61K31/506 ; A61K31/444 ; A61K31/337 ; A61K39/395 ; A61K33/24 ; A61K31/282 ; A61K31/513 ; A61K31/664 ; A61K31/427 ; A61K31/573 ; A61K31/565 ; A61K31/704 ; A61K31/7076 ; A61K31/437
摘要：
The present invention relates to triazolopyridine compounds of general formula (I) which are Monopolar Spindle 1 kinase (Mps-1 or TTK) inhibitors in which R1, R2, R3, R4, and R5 are as given in the description and in the claims, to methods of preparing said compounds, to pharmaceutical compositions and combinations comprising said compounds, to the use of said compounds for manufacturing a pharmaceutical composition for the treatment or prophylaxis of proliferative diseases, as well as to intermediate compounds useful in the preparation of said compounds.
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