发明申请
- 专利标题: BIARYL DERIVATIVES AS BROMODOMAIN INHIBITORS
- 专利标题(中): BIARYL衍生物作为BROMODOMAIN抑制剂
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申请号: US14085544申请日: 2013-11-20
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公开(公告)号: US20140140956A1公开(公告)日: 2014-05-22
- 发明人: David John Fairfax , Gregory Scott Martin , John Frederick Quinn , Bryan Cordell Duffy , Gregory Steven Wagner , Peter Ronald Young
- 申请人: David John Fairfax , Gregory Scott Martin , John Frederick Quinn , Bryan Cordell Duffy , Gregory Steven Wagner , Peter Ronald Young
- 申请人地址: CA Calgary
- 专利权人: RVX Therapeutics Inc.
- 当前专利权人: RVX Therapeutics Inc.
- 当前专利权人地址: CA Calgary
- 主分类号: C07D239/91
- IPC分类号: C07D239/91 ; A61K31/5377 ; A61K31/517 ; C07D401/14 ; C07D401/04 ; C07D409/12 ; A61K45/06 ; C07D401/12 ; A61K31/4725
摘要:
The present disclosure relates to compounds, which are useful for inhibition of BET protein function by binding to bromodomains, and their use in therapy.
公开/授权文献
- US09765039B2 Biaryl derivatives as bromodomain inhibitors 公开/授权日:2017-09-19
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