Invention Application
US20160039813A1 PROCESS FOR THE PREPARATION OF 4-(8-(2-CHLOROPHENOXY)-[1,2,4]TRIAZOLO[4,3-A]PYRIDIN-3-YL)BICYCLO[2.2.1]HEPTAN-1-OL AND NOVEL INTERMEDIATES THEREFOR
有权
制备4-（8-（2-氯苯氧基） - [1,2,4]三唑并[4,3-A]吡啶-3-基）双氰胺[2.2.1]庚烷-1-醇和新的方法 其中间性
![PROCESS FOR THE PREPARATION OF 4-(8-(2-CHLOROPHENOXY)-[1,2,4]TRIAZOLO[4,3-A]PYRIDIN-3-YL)BICYCLO[2.2.1]HEPTAN-1-OL AND NOVEL INTERMEDIATES THEREFOR](/docs/US/2016-02-11/US20160039813A1/abs.jpg.600x600.jpg)
- Patent Title: PROCESS FOR THE PREPARATION OF 4-(8-(2-CHLOROPHENOXY)-[1,2,4]TRIAZOLO[4,3-A]PYRIDIN-3-YL)BICYCLO[2.2.1]HEPTAN-1-OL AND NOVEL INTERMEDIATES THEREFOR
- Patent Title (中): 制备4-（8-（2-氯苯氧基） - [1,2,4]三唑并[4,3-A]吡啶-3-基）双氰胺[2.2.1]庚烷-1-醇和新的方法 其中间性
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Application No.: US14817352Application Date: 2015-08-04
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Publication No.: US20160039813A1Publication Date: 2016-02-11
- Inventor: Xinhua Qian , Keming Zhu , Joerg Deerberg , Wendy Wangying Yang , Kana Yamamoto , Matthew R. Hickey
- Applicant: BRISTOL-MYERS SQUIBB COMPANY
- Main IPC: C07D471/04
- IPC: C07D471/04 ; C07C51/29 ; C07D213/77 ; C07C29/00 ; C07C35/29 ; C07C61/13
![PROCESS FOR THE PREPARATION OF 4-(8-(2-CHLOROPHENOXY)-[1,2,4]TRIAZOLO[4,3-A]PYRIDIN-3-YL)BICYCLO[2.2.1]HEPTAN-1-OL AND NOVEL INTERMEDIATES THEREFOR](/abs-image/US/2016/02/11/US20160039813A1/abs.jpg.150x150.jpg)
Abstract:
A process is provided for preparing 4-(8-(2-chlorophenoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)bicyclo[2.2.1]heptan-1-ol and novel intermediates used in the process. The compound is a 11-beta hydroxysteroid dehydrogenase type I inhibitor which exhibits activity in the treatment of various metabolic diseases.
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