发明授权
- 专利标题: Pyrrolealdehydes, their preparation and their use
- 专利标题(中): 吡咯醛,其制备及其用途
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申请号: US485277申请日: 1990-02-26
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公开(公告)号: US5043348A公开(公告)日: 1991-08-27
- 发明人: Gerhard Zoller , Rudi Beyerle , Ursula Schindler
- 申请人: Gerhard Zoller , Rudi Beyerle , Ursula Schindler
- 申请人地址: DEX
- 专利权人: Cassella Aktiengesellschaft
- 当前专利权人: Cassella Aktiengesellschaft
- 当前专利权人地址: DEX
- 优先权: DEX371725 19870424
- 主分类号: C07D207/32
- IPC分类号: C07D207/32 ; C07D207/333 ; C07D403/06
摘要:
Pyrrolealdehydes of the formula I ##STR1## wherein R and R.sup.1 independently of one another denote hydrogen or alkyl with 1 to 4 C atoms, R.sup.2 denotes alkyl, which is substituted by acylamino of the formula II ##STR2## wherein X stands for an oxygen or sulphur atom and R.sup.3 denotes hydrogen, optionally substituted alkyl or alkylamino, cycloalkyl with 5 to 7 C atoms, optionally substituted phenyl, an amino group or an optionally substituted phenylamio group, and pharmaceutically acceptable acid addition salts thereof, and wherein R.sup.3 cannot represent hydrogen if R and R.sup.1 denote hydrogen and the pyrrole ring is formylated in the 3-position, their preparation and their use.