- 专利标题: Microbicidal compositions
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申请号: US537196申请日: 1990-06-12
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公开(公告)号: US5068359A公开(公告)日: 1991-11-26
- 发明人: Alica Huxley , Walter Kunz , Peter Ackermann , Marius Sutter
- 申请人: Alica Huxley , Walter Kunz , Peter Ackermann , Marius Sutter
- 申请人地址: NY Ardsley
- 专利权人: Ciba-Geigy Corporation
- 当前专利权人: Ciba-Geigy Corporation
- 当前专利权人地址: NY Ardsley
- 优先权: CHX2229/89 19890620
- 主分类号: A01N43/12
- IPC分类号: A01N43/12 ; A01N43/36 ; C07D307/79 ; C07D333/54 ; C07D333/62 ; C07D405/04 ; C07D409/04
摘要:
Novel benzothiophene and benzofuran derivatives of the general formula I ##STR1## wherein X is oxygen or sulfur, R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 haloalkyl, R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 haloalkyl, R.sub.3 is hydrogen, C.sub.1 -C.sub.4 alkyl or halogen and R is a 4-cyano-3-pyrrole radical of which the N atom carries one of the following substituents:A: hydrogen or CO--R.sub.4 in which R.sub.4 is unsubstituted C.sub.1 C.sub.6 alkyl or C.sub.1 -C.sub.6 alkyl substituted by halogen or by C.sub.1 -C.sub.3 alkoxy; C.sub.3 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl, unsubstituted C.sub.1 -C.sub.6 alkoxy or C.sub.1 -C.sub.6 alkoxy substituted by halogen or by C.sub.1 -C.sub.3 alkoxy; C.sub.3 -C.sub.6 alkenyloxy, C.sub.3 -C.sub.6 cycloalkyl or tetrahydrofur2-yl;B: S-R.sub.5 in which R.sub.5 is C.sub.1 -C.sub.3 haloalkyl;C: CH(Y)R.sub.6 in which R.sub.6 is hydrogen or C.sub.1 -C.sub.8 haloalkyl and Y is hydroxy, halogen or OC(O)R.sub.7 in which R.sub.7 is C.sub.1 -C.sub.8 alkyl, C.sub.1 -C.sub.8 haloalkyl, C.sub.2 -C.sub.6 -alkenyl, 2-tetrahydrofuryl, 2-tetrahydropyranyl or C.sub.1 -C.sub.6 alkoxycarbonyl;D: CH.sub.2 -Z in which Z is one of the groups ##STR2## wherein R.sub.8 and R.sub.9 are each, independently of the other, hydrogen, unsubstituted C.sub.1 -C.sub.6 alkyl or C.sub.1 -C.sub.6 alkyl substituted by cyano or by C.sub.1 -C.sub.6 alkoxycarbonyl; C.sub.3 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl, C.sub.3 -C.sub.7 cycloalkyl, unsubstituted phenyl or phenyl substituted by halogen, by C.sub.1 -C.sub.6 alkyl, by C.sub.1 -C.sub.6 haloalkyl and/or by C.sub.1 -C.sub.6 alkoxy, with the proviso that only R.sub.8 or R.sub.9 may be hydrogen; R.sub.10 and R.sub.11 are each, independently of the other, hydrogen, C.sub.1 -C.sub.6 alkyl or C.sub.1 -C.sub.6 alkoxycarbonyl; R.sub.12 and R.sub.13 are each, independently of the other, hydrogen, C.sub.1 -C.sub.6 alkyl or C.sub.1 -C.sub.6 alkoxycarbonyl; and R.sub.15 is oxygen, sulfur, >C.dbd.0 or >N--R.sub.14, wherein R.sub.14 is hydrogen, C.sub.1 -C.sub.6 alkyl, formyl, C.sub.1 -C.sub.6 alkanoyl or C.sub.1 -C.sub.6 alkoxycarbonyl; and n is one of the numbers 0 or 1.The novel active ingredients serve to control harmful microorganisms, especially phytophathogenic fungi. They can be used together with suitable formulation adjuvants in the form of compositions, and are suitable also for preventing attack on cultivated plants by harmful microorganisms.
公开/授权文献
- US6166259A Process for preparing a 1,1,1-trifluoro-2-aminoalkane 公开/授权日:2000-12-26