发明授权
- 专利标题: Process for the preparation of clausenamide and neoclausenamide, and derivatives thereof
- 专利标题(中): 制备杀虫剂和新西兰药物的方法及其衍生物
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申请号: US566731申请日: 1990-08-13
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公开(公告)号: US5132433A公开(公告)日: 1992-07-21
- 发明人: Liang Huang , Geng-tao Liu
- 申请人: Liang Huang , Geng-tao Liu
- 申请人地址: DEX Leverkusen CNX Beijing
- 专利权人: Bayer Aktiengesellschaft,Chinese Academy of Medical Sciences
- 当前专利权人: Bayer Aktiengesellschaft,Chinese Academy of Medical Sciences
- 当前专利权人地址: DEX Leverkusen CNX Beijing
- 优先权: DEX3927370 19890819
- 主分类号: A61K31/40
- IPC分类号: A61K31/40 ; A61K31/4015 ; A61P25/28 ; C07B53/00 ; C07D207/26 ; C07D207/273 ; C07D303/48
摘要:
A process for the preparation of compound of the formula ##STR1## in which R.sup.1 --represents ##STR2## and R.sup.2 --represents hydrogen, fluorine, chlorine or bromine. Comprising cyclizing compounds of the formula ##STR3## and, in a further step, either a) reducing stereo-specifically to give compounds of the formula in which R.sup.1 represents ##STR4## or b), to give compounds of the formula in which R.sup.1 represents ##STR5## or by c) forming compounds of the formula ##STR6## followed by stereoselective reduction to give compounds in which R.sup.1 represents ##STR7##
公开/授权文献
- US4652949A Magnetic disk loading/ejecting apparatus 公开/授权日:1987-03-24