发明授权
US5254560A 2-piperidinylpyrimidine-4-carboxamide derivatives, and their use in
therapeutics
失效
2-哌啶基嘧啶-4-甲酰胺衍生物及其在治疗中的用途
- 专利标题： 2-piperidinylpyrimidine-4-carboxamide derivatives, and their use in therapeutics
- 专利标题（中）： 2-哌啶基嘧啶-4-甲酰胺衍生物及其在治疗中的用途
-
申请号： US904061申请日： 1992-06-26
-
公开(公告)号： US5254560A公开(公告)日： 1993-10-19
- 发明人: Pascal George , Christian Maloizel , Benoit Marabout , Jean-Pierre Merly
- 申请人： Pascal George , Christian Maloizel , Benoit Marabout , Jean-Pierre Merly
- 申请人地址： FRX Le Plessis Robinson
- 专利权人： Synthelabo
- 当前专利权人： Synthelabo
- 当前专利权人地址： FRX Le Plessis Robinson
- 优先权： FRX9107938 19910627; FRX9206004 19920518
- 主分类号： A61K31/505
- IPC分类号： A61K31/505 ; A61P13/02 ; A61P15/00 ; A61P43/00 ; C07D239/42 ; C07D295/12 ; C07D401/04 ; C07D401/12
摘要：
A compound which is a carboxamide derivative of general formula (I) ##STR1## in which R represents a hydrogen atom, a methyl group or a phenoxyalkyl group of general formula ##STR2## in which X represents one or more substituents independently chosen from hydrogen, fluorine, chlorine, methyl, 1-methylethyl and methoxy andn is 2 or 3,m is 0 or 1 andp is 1 or 2 such that m+p=2q is 0 or 1, andR.sub.1 represents a hydrogen atom or a methyl group,or a pharmaceutically acceptable acid addition salt thereof. Process for their preparation and their therapeutic use.
公开/授权文献
信息查询
