发明授权
US5326760A Aminobutanoic acid compounds having metalloprotease inhibiting properties
失效
具有金属蛋白酶抑制性质的氨基丁酸化合物
- 专利标题: Aminobutanoic acid compounds having metalloprotease inhibiting properties
- 专利标题(中): 具有金属蛋白酶抑制性质的氨基丁酸化合物
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申请号: US31439申请日: 1993-03-15
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公开(公告)号: US5326760A公开(公告)日: 1994-07-05
- 发明人: Andrew B. McElroy , Peter J. Brown , David H. Drewry , James M. Salovich , Frank J. Schoenen
- 申请人: Andrew B. McElroy , Peter J. Brown , David H. Drewry , James M. Salovich , Frank J. Schoenen
- 申请人地址: NC Research Triangle Park
- 专利权人: Glaxo, Inc.
- 当前专利权人: Glaxo, Inc.
- 当前专利权人地址: NC Research Triangle Park
- 主分类号: C07C237/06
- IPC分类号: C07C237/06 ; C07D209/48 ; C07D209/66 ; C07D213/40 ; C07D401/12 ; C07D401/14 ; C07D403/12 ; C07D405/12 ; C07D409/12 ; C07D417/12 ; C07D453/02 ; C07D487/04 ; C07F7/18 ; A61K31/395 ; A61K31/40
摘要:
Aminobutanoic acids of the following formula (I): ##STR1## where R.sup.1 -R.sup.5 are a variety of substituents, novel intermediates, a pharmaceutical composition for treating inflammatory diseases, demyelinating diseases, and tumor metastasis, methods for such treatment and processes for preparing compounds of formula (I).
公开/授权文献
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