发明授权
US5792788A Substituted thiophenesulfonylureas and -thioureas, processes for their
preparation, their use as a medicament or diagnostic, and medicament
containing them
失效
取代的噻吩磺酰脲和硫脲，其制备方法，它们作为药物或诊断剂的用途，以及含有它们的药物
- 专利标题： Substituted thiophenesulfonylureas and -thioureas, processes for their preparation, their use as a medicament or diagnostic, and medicament containing them
- 专利标题（中）： 取代的噻吩磺酰脲和硫脲，其制备方法，它们作为药物或诊断剂的用途，以及含有它们的药物
-
申请号： US593621申请日： 1996-01-30
-
公开(公告)号： US5792788A公开(公告)日： 1998-08-11
- 发明人: Heinrich Englert , Jens Hartung , Peter Crause , Dieter Mania , Heinz Gogelein , Joachim Kaiser
- 申请人： Heinrich Englert , Jens Hartung , Peter Crause , Dieter Mania , Heinz Gogelein , Joachim Kaiser
- 申请人地址： DEX Frankfurt am Main
- 专利权人： Hoechst Aktiengesellschaft
- 当前专利权人： Hoechst Aktiengesellschaft
- 当前专利权人地址： DEX Frankfurt am Main
- 优先权： DEX19503136.9 19950201
- 主分类号： A61K31/38
- IPC分类号： A61K31/38 ; A61K31/381 ; A61K31/64 ; A61P9/00 ; A61P9/04 ; A61P9/06 ; A61P9/10 ; A61P43/00 ; C07C335/00 ; C07D333/34 ; C07D333/32
摘要：
Substituted thiophenesulfonylureas and -thioureas I ##STR1## wherein R(1) is selected from the group consisting of hydrogen, halogen, alkyl having 1 or 2 carbon atoms, alkoxy having 1 or 2 carbon atoms, mercaptoalkyl having 1 or 2 carbon atoms, fluoroalkoxy having 1 or 2 carbon atoms, and fluoroalkyl having 1 or 2 carbon atoms; R(2) is selected from the group consisting of hydrogen, alkyl having 1 or 2 carbon atoms such as methyl, alkoxy having 1 or 2 carbon atoms, and trifluoromethyl; X is selected from the group consisting of oxygen (compounds Ia) or sulfur (compounds Ib); Y and Z are identical or different and are selected from the group consisting of hydrogen, F, Cl, Br, I, alkyl having 1 or 2 carbon atoms and alkoxy having 1 or 2 carbon atoms.
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