Invention Grant
- Patent Title: Heterocyclic substituted piperazinone derivatives
- Patent Title (中): 杂环取代的哌嗪酮衍生物
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Application No.: US67386Application Date: 1998-04-27
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Publication No.: US5864045APublication Date: 1999-01-26
- Inventor: Timothy P. Burkholder , Elizabeth M. Kudlacz , Tieu-Binh Le
- Applicant: Timothy P. Burkholder , Elizabeth M. Kudlacz , Tieu-Binh Le
- Applicant Address: OH Cincinnati
- Assignee: Hoechst Marion Roussel, Inc.
- Current Assignee: Hoechst Marion Roussel, Inc.
- Current Assignee Address: OH Cincinnati
- Main IPC: A61K31/495
- IPC: A61K31/495 ; A61P11/00 ; A61P43/00 ; C07D209/04 ; C07D209/08 ; C07D209/20 ; C07D403/06 ; C07D403/14
Abstract:
The present invention relates to substituted piperazinone derivatives of formula (1) or stereoisomers, or pharmaceutically acceptable salts thereof and their use as tachykinin receptor antagonists. Such antagonists are useful in the treatment of tachykinin-mediated diseases and conditions disclosed herein including: asthma, cough, and bronchitis. The present invention also relates to intermediates useful in the preparation of compounds of formula (1).
Public/Granted literature
- USD392600S Motorcycle body Public/Granted day:1998-03-24
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