发明授权
US6004975A Bicyclolactam compounds, use thereof and intermediates for preparing
thereof
失效
双环内酰胺化合物，其用途及其制备中间体
- 专利标题： Bicyclolactam compounds, use thereof and intermediates for preparing thereof
- 专利标题（中）： 双环内酰胺化合物，其用途及其制备中间体
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申请号： US908601申请日： 1997-08-08
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公开(公告)号： US6004975A公开(公告)日： 1999-12-21
- 发明人: Junji Yamamoto , Takashi Arima , Nobuo Kasahara , Masato Nanri , Kazuo Ogawa , Ichiro Yamawaki , Manabu Kaneda
- 申请人： Junji Yamamoto , Takashi Arima , Nobuo Kasahara , Masato Nanri , Kazuo Ogawa , Ichiro Yamawaki , Manabu Kaneda
- 申请人地址： JPX Tokyo
- 专利权人： Taiho Pharmaceutical Company Limited
- 当前专利权人： Taiho Pharmaceutical Company Limited
- 当前专利权人地址： JPX Tokyo
- 优先权： JPX6-83934 19940328; JPX7-170329 19950612; JPX7-274654 19950927
- 主分类号： A61K31/40
- IPC分类号： A61K31/40 ; A61K31/445 ; A61K31/47 ; A61K31/55 ; C07D215/22 ; C07D215/227 ; C07D221/16 ; C07D221/04 ; A61K31/435
摘要：
A bicyclolactam compound of the formula (1) is disclosed, which has an excellent anxiolytic effect, is high in safety, and is useful as an effective component of medicinals which are greatly diminished in side effects such as hypnotic, muscle relaxant and sedative effects ##STR1## A bicyclolactam derivative represented by the following formula (1) is also disclosed, and is useful as an effective component of an anxiolytic agent ##STR2## .