发明授权
US06414160B1 Process for producing 4-alkoxycarbonyl-2-oxazolidinone compound
失效
制备4-烷氧基羰基-2-恶唑烷酮化合物的方法
- 专利标题: Process for producing 4-alkoxycarbonyl-2-oxazolidinone compound
- 专利标题(中): 制备4-烷氧基羰基-2-恶唑烷酮化合物的方法
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申请号: US09480558申请日: 2000-01-10
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公开(公告)号: US06414160B1公开(公告)日: 2002-07-02
- 发明人: Hiroyuki Miyata , Nobuya Satake , Takashi Honma , Kikuo Ataka
- 申请人: Hiroyuki Miyata , Nobuya Satake , Takashi Honma , Kikuo Ataka
- 优先权: JP9-185150 19970710
- 主分类号: C07D26338
- IPC分类号: C07D26338
摘要:
The present invention relates to a process for producing 4-alkoxycarbonyl-2-oxazolidinone compound represented by the formula (III): wherein R1 represents H, an alkyl group, an cycloalkyl group, an alkenyl group or a phenyl group, R2 represents H, an alkyl group, a phenyl group or an alkenyl group, R3 represents an alkyl group, a cycloalkyl group, an alkenyl group, or a phenyl group, and R4 represents H, an alkyl group, an alkenyl group, acycloalkyl group, alkynyl group, an aryl group, a 5- or 6-membered heteroaromatic ring group, an alkoxycarbonyl group, an acetyl group or a benzoyl group, which comprises reacting a 5-alkoxy-2(3H)oxazolone compound represented by the formula (I): wherein R1, R2 and R3 have the same meanings as defined above, and an aldehyde compound represented by the formula (II): R4CHO (II) wherein R4 has the same meaning as defined above, in the presence of a Lewis acid catalyst.