发明授权
US06472538B1 Method for producing 1-substituted 5-hydroxypyrazoles 失效
1-取代的5-羟基吡唑的制备方法

  • 专利标题: Method for producing 1-substituted 5-hydroxypyrazoles
  • 专利标题(中): 1-取代的5-羟基吡唑的制备方法
  • 申请号: US09830350
    申请日: 2001-04-25
  • 公开(公告)号: US06472538B1
    公开(公告)日: 2002-10-29
  • 发明人: Norbert GötzRoland GötzMichael Rack
  • 申请人: Norbert GötzRoland GötzMichael Rack
  • 优先权: DE19851100 19981105; DE19910505 19990310
  • 主分类号: C07D23120
  • IPC分类号: C07D23120
Method for producing 1-substituted 5-hydroxypyrazoles
摘要:
A process for preparing compounds of the formula I in which R1 is hydrogen, an aliphatic group having 1-8 carbon atoms, C1-C6-alkoxycarbonyl, C1-C6-alkylthiocarbonyl or a cyclic ring system having 3-14 ring atoms, and R2 is hydrogen, an aliphatic group having 1-8 carbon atoms, or R1 and R2 together with the carbon atom to which they are bound form a cyclic or bicyclic ring system having 3-14 ring atoms, comprises the preparation of compounds of the formula II  in which R3 and R4 are readily detachable groups and R1 and R2 are as defined above, as starting materials or intermediates and the cyclization of these under suitable reaction conditions to give compounds of the formula I.
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