Invention Grant
- Patent Title: Preparation of isoxazolin-3-ylacylbenzenes
- Patent Title (中): 异恶唑啉-3-基酰基苯的制备
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Application No.: US10180608Application Date: 2002-06-27
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Publication No.: US06608209B2Publication Date: 2003-08-19
- Inventor: Joachim Rheinheimer , Wolfgang von Deyn , Joachim Gebhardt , Michael Rack , Rene Lochtman , Norbert Götz , Michael Keil , Matthias Witschel , Helmut Hagen , Ulf Misslitz , Ernst Baumann
- Applicant: Joachim Rheinheimer , Wolfgang von Deyn , Joachim Gebhardt , Michael Rack , Rene Lochtman , Norbert Götz , Michael Keil , Matthias Witschel , Helmut Hagen , Ulf Misslitz , Ernst Baumann
- Priority: DE19820722 19980511; DE19852095 19981112
- Main IPC: C07D26102
- IPC: C07D26102

Abstract:
A process is described for preparing isoxazoles of the formula I wherein R1 is hydrogen, C1-C6-alkyl, R2 is C1-C6-alkyl, R3, R4, R5 are hydrogen, C1-C6-alkyl, or R4 and R5 together form a bond, R6 is a heterocyclic ring, n is 0, 1 or 2; in which an intermediate of the formula VI is prepared, followed by halogenation, thiomethylation, oxidation and acylation to give compounds of formula I. Novel intermediates for preparing the intermediates are described.
Public/Granted literature
- US20030018200A1 Preparation of isoxazolin-3-ylacylbenzenes Public/Granted day:2003-01-23
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