Invention Grant
US06608209B2 Preparation of isoxazolin-3-ylacylbenzenes 有权
异恶唑啉-3-基酰基苯的制备

Preparation of isoxazolin-3-ylacylbenzenes
Abstract:
A process is described for preparing isoxazoles of the formula I wherein R1 is hydrogen, C1-C6-alkyl, R2 is C1-C6-alkyl, R3, R4, R5 are hydrogen, C1-C6-alkyl, or R4 and R5 together form a bond, R6 is a heterocyclic ring, n is 0, 1 or 2; in which an intermediate of the formula VI  is prepared, followed by halogenation, thiomethylation, oxidation and acylation to give compounds of formula I. Novel intermediates for preparing the intermediates are described.
Public/Granted literature
Information query
Patent Agency Ranking
0/0