Invention Grant
- Patent Title: Pyridopyrimidine derivatives as 5-HT6 antagonists
- Patent Title (中): 吡啶并嘧啶衍生物作为5-HT6拮抗剂
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Application No.: US10620240Application Date: 2003-07-15
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Publication No.: US06875771B2Publication Date: 2005-04-05
- Inventor: Yong-Jin Wu , Shuanghua Hu , Paul M. Scola , Yazhong Huang , Katharine A. Grant-Young
- Applicant: Yong-Jin Wu , Shuanghua Hu , Paul M. Scola , Yazhong Huang , Katharine A. Grant-Young
- Applicant Address: US NJ Princeton
- Assignee: Bristol-Myers Squibb Company
- Current Assignee: Bristol-Myers Squibb Company
- Current Assignee Address: US NJ Princeton
- Agent Aldo A. Algieri
- Main IPC: A61K31/519
- IPC: A61K31/519 ; C07D471/04 ; C07D471/14 ; C07D487/02

Abstract:
Novel pyridopyrimidine derivatives which have a binding affinity for the human 5-HT6 receptor and, therefore, are useful in treating disorders responsive to antagonism of the 5-HT6 receptor such as psychosis, schizophrenia, manic depression, depression, neurological disorder, memory disorder, Parkinson's disease, amyotrophic lateral sclerosis, Alzheimer's disease and Huntington's chorea.
Public/Granted literature
- US20040019064A1 Pyridopyrimidine derivatives as 5-HT6 antagonists Public/Granted day:2004-01-29
Information query
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