Invention Grant
US07405305B2 Pyrrole-2, 5dione derivatives and their used as GSK-3 inhibitors
失效
吡咯-2,5-二酮衍生物,用作GSK-3抑制剂
- Patent Title: Pyrrole-2, 5dione derivatives and their used as GSK-3 inhibitors
- Patent Title (中): 吡咯-2,5-二酮衍生物,用作GSK-3抑制剂
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Application No.: US10506029Application Date: 2003-03-05
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Publication No.: US07405305B2Publication Date: 2008-07-29
- Inventor: Pamela Ann Albaugh , Jochen Ammenn , Timothy Paul Burkholder , Joshua Ryan Clayton , Scott Eugene Conner , Brian Eugene Cunningham , Thomas Albert Engler , Kelly Wayne Furness , James Robert Henry , Sushant Malhotra , Mark Joseph Tebbe , Guoxin Zhu , YiHong Li , Brian Raymond Berridge , Charles Edward Ruegg , John Morris Sullivan
- Applicant: Pamela Ann Albaugh , Jochen Ammenn , Timothy Paul Burkholder , Joshua Ryan Clayton , Scott Eugene Conner , Brian Eugene Cunningham , Thomas Albert Engler , Kelly Wayne Furness , James Robert Henry , Sushant Malhotra , Mark Joseph Tebbe , Guoxin Zhu , YiHong Li , Brian Raymond Berridge , Charles Edward Ruegg , John Morris Sullivan
- Applicant Address: US IN Indianapolis
- Assignee: Eli Lilly and Company
- Current Assignee: Eli Lilly and Company
- Current Assignee Address: US IN Indianapolis
- Agent Robert D. Titus
- International Application: PCT/US03/05052 WO 20030305
- International Announcement: WO03/076398 WO 20030918
- Main IPC: C07D209/12
- IPC: C07D209/12 ; C07D207/24 ; C07D211/06

Abstract:
The present invention provides kinase inhibitors of Formula (I)
Public/Granted literature
- US20050288321A1 Kinase inhibitors Public/Granted day:2005-12-29
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