-
公开(公告)号:US08058425B2
公开(公告)日:2011-11-15
申请号:US13100618
申请日:2011-05-04
Applicant: Thomas Albert Engler , Timothy Paul Burkholder , Joshua Ryan Clayton , Clive Gideon Diefenbacher , Kelly Wayne Furness , James Robert Henry , Yihong Li , Sushant Malhotra , Angela Lynn Marquart , Johnathan Alexander McLean , David Mendel , Jon Kevin Reel , Brian Raymond Berridge , Charles Edward Ruegg , John Morris Sullivan
Inventor: Thomas Albert Engler , Timothy Paul Burkholder , Joshua Ryan Clayton , Clive Gideon Diefenbacher , Kelly Wayne Furness , James Robert Henry , Yihong Li , Sushant Malhotra , Angela Lynn Marquart , Johnathan Alexander McLean , David Mendel , Jon Kevin Reel , Brian Raymond Berridge , Charles Edward Ruegg , John Morris Sullivan
IPC: A61P25/08 , A61K31/55 , C07D487/06
CPC classification number: C07D471/06 , C07D487/06
Abstract: The present invention provides kinase inhibitors of Formula I.
Abstract translation: 本发明提供式的激酶抑制剂。
-
2.Pyrrole-2, 5dione derivatives and their used as GSK-3 inhibitors 失效
Title translation: 吡咯-2,5-二酮衍生物,用作GSK-3抑制剂公开(公告)号:US07405305B2
公开(公告)日:2008-07-29
申请号:US10506029
申请日:2003-03-05
Applicant: Pamela Ann Albaugh , Jochen Ammenn , Timothy Paul Burkholder , Joshua Ryan Clayton , Scott Eugene Conner , Brian Eugene Cunningham , Thomas Albert Engler , Kelly Wayne Furness , James Robert Henry , Sushant Malhotra , Mark Joseph Tebbe , Guoxin Zhu , YiHong Li , Brian Raymond Berridge , Charles Edward Ruegg , John Morris Sullivan
Inventor: Pamela Ann Albaugh , Jochen Ammenn , Timothy Paul Burkholder , Joshua Ryan Clayton , Scott Eugene Conner , Brian Eugene Cunningham , Thomas Albert Engler , Kelly Wayne Furness , James Robert Henry , Sushant Malhotra , Mark Joseph Tebbe , Guoxin Zhu , YiHong Li , Brian Raymond Berridge , Charles Edward Ruegg , John Morris Sullivan
IPC: C07D209/12 , C07D207/24 , C07D211/06
CPC classification number: C07D451/04 , C07D401/14 , C07D403/04 , C07D403/14 , C07D405/14 , C07D471/04 , C07D491/04
Abstract: The present invention provides kinase inhibitors of Formula (I)
Abstract translation: 本发明提供式(I)的激酶抑制剂,
-
公开(公告)号:US20110294792A1
公开(公告)日:2011-12-01
申请号:US13206057
申请日:2011-08-09
Applicant: Thomas Albert Engler , Timothy Paul Burkholder , Joshua Ryan Clayton , Clive Gideon Diefenbacher , Kelly Wayne Furness , James Robert Henry , Yihong Li , Sushant Malhotra , Angela Lynn Marquart , Johnathan Alexander McLean , David Mendel , Jon Kevin Reel , Brian Raymond Berridge , Charles Edward Ruegg , John Morris Sullivan
Inventor: Thomas Albert Engler , Timothy Paul Burkholder , Joshua Ryan Clayton , Clive Gideon Diefenbacher , Kelly Wayne Furness , James Robert Henry , Yihong Li , Sushant Malhotra , Angela Lynn Marquart , Johnathan Alexander McLean , David Mendel , Jon Kevin Reel , Brian Raymond Berridge , Charles Edward Ruegg , John Morris Sullivan
IPC: A61K31/551 , A61P19/08 , C07D487/04
CPC classification number: C07D471/06 , C07D487/06
Abstract: The present invention provides kinase inhibitors of Formula I.
-
公开(公告)号:US20110207721A1
公开(公告)日:2011-08-25
申请号:US13100618
申请日:2011-05-04
Applicant: Thomas Albert Engler , Timothy Paul Burkholder , Joshua Ryan Clayton , Clive Gideon Diefenbacher , Kelly Wayne Furness , James Robert Henry , Yihong Li , Sushant Malhotra , Angela Lynn Marquart , Johnathan Alexander McLean , David Mendel , Jon Kevin Reel , Brian Raymond Berridge , Charles Edward Ruegg , John Morris Sullivan
Inventor: Thomas Albert Engler , Timothy Paul Burkholder , Joshua Ryan Clayton , Clive Gideon Diefenbacher , Kelly Wayne Furness , James Robert Henry , Yihong Li , Sushant Malhotra , Angela Lynn Marquart , Johnathan Alexander McLean , David Mendel , Jon Kevin Reel , Brian Raymond Berridge , Charles Edward Ruegg , John Morris Sullivan
IPC: A61K31/5517 , C07D487/04 , A61P3/10 , A61P25/28
CPC classification number: C07D471/06 , C07D487/06
Abstract: The present invention provides kinase inhibitors of Formula I.
Abstract translation: 本发明提供式I的激酶抑制剂。
-
-
-