发明授权
US07465735B2 5-Phenypyrimidines their preparation compositions comprising them and their use
失效
5-苯氧基嘧啶制备它们的组合物及其用途
- 专利标题: 5-Phenypyrimidines their preparation compositions comprising them and their use
- 专利标题(中): 5-苯氧基嘧啶制备它们的组合物及其用途
-
申请号: US10495280申请日: 2002-11-15
-
公开(公告)号: US07465735B2公开(公告)日: 2008-12-16
- 发明人: Andreas Gypser , Thomas Grote , Anja Schwögler , Joachim Rheinheimer , Frank Schieweck , Jordi Tormo i Blasco , Ingo Rose , Peter Schäfer , Markus Gewehr , Wassilios Grammenos , Bernd Müller , Eberhard Ammermann , Siegfried Strathmann , Gisela Lorenz , Reinhard Stierl
- 申请人: Andreas Gypser , Thomas Grote , Anja Schwögler , Joachim Rheinheimer , Frank Schieweck , Jordi Tormo i Blasco , Ingo Rose , Peter Schäfer , Markus Gewehr , Wassilios Grammenos , Bernd Müller , Eberhard Ammermann , Siegfried Strathmann , Gisela Lorenz , Reinhard Stierl
- 申请人地址: DE Ludwigshafen
- 专利权人: BASF Aktiengesellschaft
- 当前专利权人: BASF Aktiengesellschaft
- 当前专利权人地址: DE Ludwigshafen
- 代理机构: Novak Druce + Quigg LLP
- 优先权: DE10156279 20011119
- 国际申请: PCT/EP02/12807 WO 20021115
- 国际公布: WO03/043993 WO 20030530
- 主分类号: C07D239/42
- IPC分类号: C07D239/42 ; C07D239/46 ; C07D239/48 ; C07D239/52 ; C07D401/12 ; C07D403/12 ; A61K31/505 ; A61K31/506 ; A01N43/54
摘要:
5-Phenylpyrimidines, their preparation, compositions comprising them and their use 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC(═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC(═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C(═O)NRaRb or —C(═O)Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
公开/授权文献
信息查询