Invention Grant
- Patent Title: Preparation of isoxazolin-3-ylacylbenzene
- Patent Title (中): 异恶唑啉-3-基酰基苯的制备
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Application No.: US11684630Application Date: 2007-03-11
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Publication No.: US07663001B2Publication Date: 2010-02-16
- Inventor: Joachim Rheinheimer , Wolfgang von Deyn , Joachim Gebhardt , Michael Rack , Rene Lochtman , Norbert Götz , Michael Keil , Matthias Witschel , Helmut Hagen , Ulf Miβlitz , Ernst Baumann
- Applicant: Joachim Rheinheimer , Wolfgang von Deyn , Joachim Gebhardt , Michael Rack , Rene Lochtman , Norbert Götz , Michael Keil , Matthias Witschel , Helmut Hagen , Ulf Miβlitz , Ernst Baumann
- Applicant Address: DE Ludwigshafen
- Assignee: BASF Aktiengesellschaft
- Current Assignee: BASF Aktiengesellschaft
- Current Assignee Address: DE Ludwigshafen
- Agency: Novak Druce + Quigg LLP
- Priority: DE19820722 19980511; DE19852095 19981112
- Main IPC: C07C239/08
- IPC: C07C239/08

Abstract:
A process is described for preparing isoxazoles of the formula I where the substituents are as defined below: R1 is hydrogen, C1-C6-alkyl, R2 is C1-C6-alkyl, R3, R4, R5 are hydrogen, C1-C6-alkyl, or R4 and R5 together form a bond, R6 is a heterocyclic ring, n is 0, 1 or 2; which comprises preparing an intermediate of the formula VI where R1, R3, R4 and R5 are as defined above, followed by halogenation, thiomethylation, oxidation and acylation to give compounds of the formula I. Also novel intermediates for preparing the compounds of the formula I and novel processes for preparing the intermediates are described.
Public/Granted literature
- US20070161800A1 Preparation of Isoxazolin-3-Ylacylbenzene Public/Granted day:2007-07-12
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