发明授权
US07846922B2 1-benzoyl substituted diazepine derivatives as selective histamine H3 receptor agonists
失效
1-苯甲酰基取代的二氮杂衍生物作为选择性组胺H3受体激动剂
- 专利标题: 1-benzoyl substituted diazepine derivatives as selective histamine H3 receptor agonists
- 专利标题(中): 1-苯甲酰基取代的二氮杂衍生物作为选择性组胺H3受体激动剂
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申请号: US10576492申请日: 2004-10-14
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公开(公告)号: US07846922B2公开(公告)日: 2010-12-07
- 发明人: Gordon Bruton , Anthony Huxley , Barry Sidney Orlek , Kishore Kalidas Rana
- 申请人: Gordon Bruton , Anthony Huxley , Barry Sidney Orlek , Kishore Kalidas Rana
- 申请人地址: GB Greenford, Middlesex
- 专利权人: Glaxo Group Limited
- 当前专利权人: Glaxo Group Limited
- 当前专利权人地址: GB Greenford, Middlesex
- 代理商 Bonnie L. Deppenbrock
- 优先权: GB0324159.3 20031015
- 国际申请: PCT/EP2004/011619 WO 20041014
- 国际公布: WO2005/040144 WO 20050506
- 主分类号: A61P25/00
- IPC分类号: A61P25/00 ; A61K31/551 ; C07D241/12 ; C07D231/14 ; C07D239/26 ; C07D237/08 ; C07D213/81 ; C07D263/32 ; C07D257/04 ; C07D295/18
摘要:
The present invention relates to novel diazepanyl derivatives of formula (I) having pharmacological activity, processes for their preparation, to compositions containing them and to their use in the treatment of neurological and psychiatric disorders.