发明授权
- 专利标题: Polymorphic forms of a GABAA agonist
- 专利标题(中): 多形态的GABAA激动剂
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申请号: US11813796申请日: 2006-01-26
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公开(公告)号: US08022084B2公开(公告)日: 2011-09-20
- 发明人: Daniel J. Kumke , Jerry A. Murry , Bryon L. Simmons , Feng Xu
- 申请人: Daniel J. Kumke , Jerry A. Murry , Bryon L. Simmons , Feng Xu
- 申请人地址: DK Valby
- 专利权人: H. Lundbeck A/S
- 当前专利权人: H. Lundbeck A/S
- 当前专利权人地址: DK Valby
- 代理机构: Fish & Richardson P.C.
- 国际申请: PCT/US2006/002809 WO 20060126
- 国际公布: WO2006/083682 WO 20060810
- 主分类号: A61K31/4355
- IPC分类号: A61K31/4355 ; C07D498/04
摘要:
The present invention is directed to novel polymorphic forms of the compound 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol hydrate (gaboxadol monohydrate). The invention is further concerned with pharmaceutical compositions containing the polymorphic forms as an active ingredient, methods for treatment of disorders susceptible to amelioration by GABAA receptor agonism with the polymorphic forms, and processes for the preparation of the polymorphic forms.
公开/授权文献
- US20080085913A1 Polymorphic Forms of a Gabaa Agonist 公开/授权日:2008-04-10