Invention Grant
US08147880B2 Polyacetylenic compounds for stimulating insulin gene exression, production and secretion
有权
用于刺激胰岛素基因表达,产生和分泌的聚乙炔化合物
- Patent Title: Polyacetylenic compounds for stimulating insulin gene exression, production and secretion
- Patent Title (中): 用于刺激胰岛素基因表达,产生和分泌的聚乙炔化合物
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Application No.: US12766895Application Date: 2010-04-25
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Publication No.: US08147880B2Publication Date: 2012-04-03
- Inventor: Wen-Chin Yang
- Applicant: Wen-Chin Yang
- Applicant Address: TW Taipei
- Assignee: Academia Sinica
- Current Assignee: Academia Sinica
- Current Assignee Address: TW Taipei
- Agency: Intellectual Property Connections, Inc.
- Agent Hsiu-Ming Saunders
- Main IPC: A61K36/00
- IPC: A61K36/00

Abstract:
This invention relates to a method of treating type II diabetes with a polyacetylenic compound of the following formula: in which R1 is H, C1-C10 alkyl, C2-C10 alkenyl, C2-C10 alkynyl, C3-C20 cycloalkyl, C3-C20 cycloalkenyl, C1-C20 heterocycloalkyl, C1-C20 heterocycloalkenyl, aryl, or heteroaryl; R2 is H or a monosaccharide residue; R3 is H or C1-C10 alkyl; m is 2, 3, or 4; n is 0, 1, 2, or 3; o is 0, 1, 2, 3, or 4; and p is 1, 2, 3, or 4.
Public/Granted literature
- US20100204166A1 POLYACETYLENIC COMPOUNDS FOR STIMULATING INSULIN GENE EXRESSION, PRODUCTION AND SECRETION Public/Granted day:2010-08-12
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