发明授权
US08524906B2 Tetrahydrothiazolopyridine inhibitors of phosphatidylinositol 3-kinase
失效
磷脂酰肌醇3-激酶的四氢噻唑并吡啶抑制剂
- 专利标题: Tetrahydrothiazolopyridine inhibitors of phosphatidylinositol 3-kinase
- 专利标题(中): 磷脂酰肌醇3-激酶的四氢噻唑并吡啶抑制剂
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申请号: US13211502申请日: 2011-08-17
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公开(公告)号: US08524906B2公开(公告)日: 2013-09-03
- 发明人: Alex Aronov , Upul Keerthi Bandarage , Kevin Michael Cottrell , Robert J. Davies , Elaine B. Krueger , Mark Willem Ledeboer , Brian Ledford , Arnaud Le Tiran , David Messersmith , Tiansheng Wang , Jinwang Xu , Yusheng Liao
- 申请人: Alex Aronov , Upul Keerthi Bandarage , Kevin Michael Cottrell , Robert J. Davies , Elaine B. Krueger , Mark Willem Ledeboer , Brian Ledford , Arnaud Le Tiran , David Messersmith , Tiansheng Wang , Jinwang Xu , Yusheng Liao
- 申请人地址: US MA Cambridge
- 专利权人: Vertex Pharmaceuticals Incorporated
- 当前专利权人: Vertex Pharmaceuticals Incorporated
- 当前专利权人地址: US MA Cambridge
- 代理商 Daniel A. Pearson
- 主分类号: A61K31/4365
- IPC分类号: A61K31/4365 ; C07D513/04
摘要:
The present invention relates to compounds useful as inhibitors of PI3K, particularly of PI3Kγ. The invention also provides pharmaceutically acceptable compositions comprising said compounds and methods of using the compositions in the treatment of various disease, conditions, or disorders.