- 专利标题: Nitrogen containing heteroaryl compounds
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申请号: US13151301申请日: 2011-06-02
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公开(公告)号: US08623866B2公开(公告)日: 2014-01-07
- 发明人: Konrad Bleicher , Alexander Flohr , Katrin Groebke Zbinden , Felix Gruber , Matthias Koerner , Bernd Kuhn , Jens-Uwe Peters , Rosa Maria Rodriguez-Sarmiento
- 申请人: Konrad Bleicher , Alexander Flohr , Katrin Groebke Zbinden , Felix Gruber , Matthias Koerner , Bernd Kuhn , Jens-Uwe Peters , Rosa Maria Rodriguez-Sarmiento
- 申请人地址: US NJ Nutley
- 专利权人: Hoffmann-La Roche Inc.
- 当前专利权人: Hoffmann-La Roche Inc.
- 当前专利权人地址: US NJ Nutley
- 优先权: EP10165427 20100609
- 主分类号: C07D239/42
- IPC分类号: C07D239/42 ; A01N43/54 ; A61K31/5355 ; C07D403/14 ; A61K31/497 ; A61P25/18
摘要:
The invention is concerned with novel nitrogen-containing heteroaryl compounds of formula (I) wherein A1, A2, R1, R2, R3, R4, R5 and R6 are as defined in the description and in the claims, as well as physiologically acceptable salts and esters thereof. These compounds inhibit PDE10A and can be used as therapeutics.
公开/授权文献
- US08703768B2 Nitrogen containing heteroaryl compounds 公开/授权日:2014-04-22
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