发明授权
- 专利标题: Chiral intermediates useful for the preparation of hydroxyphosphine ligands
- 专利标题(中): 用于制备羟基膦配体的手性中间体
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申请号: US13882580申请日: 2011-11-01
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公开(公告)号: US08993788B2公开(公告)日: 2015-03-31
- 发明人: Jaidev Rajnikant Shroff , Vikram Rajnikant Shroff , Birja Shanker
- 申请人: Jaidev Rajnikant Shroff , Vikram Rajnikant Shroff , Birja Shanker
- 申请人地址: IN Mumbai, Maharashtra
- 专利权人: UPL Limited
- 当前专利权人: UPL Limited
- 当前专利权人地址: IN Mumbai, Maharashtra
- 代理机构: Merchant & Gould P.C.
- 优先权: IN3045/MUM/2010 20101102; IN3046/MUM/2010 20101102
- 国际申请: PCT/IB2011/002587 WO 20111101
- 国际公布: WO2012/059807 WO 20120510
- 主分类号: C07C31/135
- IPC分类号: C07C31/135 ; C07F9/50 ; C07C43/21 ; C07D309/12 ; C07F7/08 ; C07C29/149 ; C07C29/64 ; C07C67/08 ; C07C67/14 ; C07D309/10 ; C07D309/30
摘要:
A compound of formula (I), wherein R1 is hydrogen or a hydroxyl protecting group; and R2 and R3 are same or different and are independently selected from halogen or —O—SO2—X; wherein X is —C1-C4 alkyl; C1-C4 alkyl substituted with one or more halogen; or substituted or unsubstituted phenyl wherein said phenyl substituent is selected from halogen, nitro and C1-C4 alkyl; provided that when R3 is bromine, X is not p-toluoyl; and a process for the preparation thereof.
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