Invention Grant
US09242976B2 Thiazolyl- or thiadiazolyl-substituted pyridyl compounds useful as kinase inhibitors
有权
可用作激酶抑制剂的噻唑基或噻二唑基取代的吡啶基化合物
- Patent Title: Thiazolyl- or thiadiazolyl-substituted pyridyl compounds useful as kinase inhibitors
- Patent Title (中): 可用作激酶抑制剂的噻唑基或噻二唑基取代的吡啶基化合物
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Application No.: US14371463Application Date: 2013-01-11
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Publication No.: US09242976B2Publication Date: 2016-01-26
- Inventor: Venkatram Reddy Paidi , Sreekantha Ratna Kumar , Abhisek Banerjee , Ramesh Sistla , Satheesh Kesavan Nair , William J. Pitts , John Hynes
- Applicant: BRISTOL-MYERS SQUIBB COMPANY
- Applicant Address: US NJ Princeton
- Assignee: Bristol-Myers Squibb Company
- Current Assignee: Bristol-Myers Squibb Company
- Current Assignee Address: US NJ Princeton
- Agent Gary D. Greenblatt
- International Application: PCT/US2013/021134 WO 20130111
- International Announcement: WO2013/106641 WO 20130718
- Main IPC: C07D417/14
- IPC: C07D417/14 ; C07D413/14 ; C07D413/04 ; C07D417/04 ; C07D471/04 ; C07D487/04

Abstract:
Compounds having the following formula (I) or an enantiomer, diastereomer or a pharmaceutically-acceptable salt thereof, wherein X is N or C—R7, are useful as kinase modulators, including IRAK-4 modulation.
Public/Granted literature
- US20150018344A1 THIAZOLYL- OR THIADIAZOLYL-SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS KINASE INHIBITORS Public/Granted day:2015-01-15
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