Invention Grant
US09580420B2 Process for the preparation of 4-(8-(2-chlorophenoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)bicyclo[2.2.1]heptan-1-ol and novel intermediates therefor
有权
制备4-（8-（2-氯苯氧基） - [1,2,4]三唑并[4,3-a]吡啶-3-基）双环[2.2.1]庚-1-醇的方法和新颖的 中间体
![Process for the preparation of 4-(8-(2-chlorophenoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)bicyclo[2.2.1]heptan-1-ol and novel intermediates therefor](/docs/US/2017-02-28/US09580420B2/abs.jpg.600x600.jpg)
- Patent Title: Process for the preparation of 4-(8-(2-chlorophenoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)bicyclo[2.2.1]heptan-1-ol and novel intermediates therefor
- Patent Title (中): 制备4-（8-（2-氯苯氧基） - [1,2,4]三唑并[4,3-a]吡啶-3-基）双环[2.2.1]庚-1-醇的方法和新颖的 中间体
-
Application No.: US14817352Application Date: 2015-08-04
-
Publication No.: US09580420B2Publication Date: 2017-02-28
- Inventor: Xinhua Qian , Keming Zhu , Joerg Deerberg , Wendy Wangying Yang , Kana Yamamoto , Matthew R. Hickey
- Applicant: BRISTOL-MYERS SQUIBB COMPANY
- Applicant Address: US NJ Princeton
- Assignee: Bristol-Meyers Squibb Company
- Current Assignee: Bristol-Meyers Squibb Company
- Current Assignee Address: US NJ Princeton
- Agent Elliott Korsen
- Main IPC: C07D213/77
- IPC: C07D213/77 ; C07C35/29 ; C07D471/04 ; C07C29/00 ; C07C51/29 ; C07C61/13
![Process for the preparation of 4-(8-(2-chlorophenoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)bicyclo[2.2.1]heptan-1-ol and novel intermediates therefor](/abs-image/US/2017/02/28/US09580420B2/abs.jpg.150x150.jpg)
Abstract:
A process is provided for preparing 4-(8-(2-chlorophenoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)bicyclo[2.2.1]heptan-1-ol and novel intermediates used in the process. The compound is a 11-beta hydroxysteroid dehydrogenase type I inhibitor which exhibits activity in the treatment of various metabolic diseases.
Public/Granted literature
Information query
IPC分类:
