Invention Grant
- Patent Title: Solid preparation
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Application No.: US15272755Application Date: 2016-09-22
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Publication No.: US09757377B2Publication Date: 2017-09-12
- Inventor: Maiko Harada , Ikurou Yamane , Masafumi Misaki
- Applicant: Takeda Pharmaceutical Company Limited
- Applicant Address: JP Osaka
- Assignee: Takeda Pharmaceutical Company Limited
- Current Assignee: Takeda Pharmaceutical Company Limited
- Current Assignee Address: JP Osaka
- Agency: Foley & Lardner LLP
- Priority: JP2012-128360 20120605
- Main IPC: A61K9/28
- IPC: A61K9/28 ; A61K31/51 ; A61K9/20 ; A61K9/16 ; A61K31/506 ; A61K31/513

Abstract:
The present invention provides a solid preparation excellent in disintegration property and preservation stability. The present invention relates to a solid preparation containing (1) 2-[[6-[(3R)-3-amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]-4-fluorobenzonitrile (compound (A)) or a salt thereof, (2) a saccharide, and (3) sodium stearyl fumarate. In addition, the present invention relates to a solid preparation containing (1) compound (A) or a salt thereof, (2) a saccharide, and (3) stearic acid or talc in a naked tablet part.
Public/Granted literature
- US20170007607A1 SOLID PREPARATION Public/Granted day:2017-01-12
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