Invention Application
- Patent Title: CONDENSED DIHYDROQUINOLINONE DERIVATIVES FOR INHIBITING MRP1
- Patent Title (中): 用于抑制MRP1的冷凝二氢喹啉酮衍生物
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Application No.: PCT/US0021980Application Date: 2000-09-22
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Publication No.: WO0127116A3Publication Date: 2001-11-22
- Inventor: BONJOUKLIAN ROSANNE , JOHNSON DOUGLAS WEBB , LANDER PETER AMBROSE , LOHMAN MARK CHRISTOPHER , PATEL VINOD FRANCIS , VEPACHEDU SREENIVASARAO , XIE YONGPING
- Applicant: LILLY CO ELI , BONJOUKLIAN ROSANNE , JOHNSON DOUGLAS WEBB , LANDER PETER AMBROSE , LOHMAN MARK CHRISTOPHER , PATEL VINOD FRANCIS , VEPACHEDU SREENIVASARAO , XIE YONGPING
- Assignee: LILLY CO ELI,BONJOUKLIAN ROSANNE,JOHNSON DOUGLAS WEBB,LANDER PETER AMBROSE,LOHMAN MARK CHRISTOPHER,PATEL VINOD FRANCIS,VEPACHEDU SREENIVASARAO,XIE YONGPING
- Current Assignee: LILLY CO ELI,BONJOUKLIAN ROSANNE,JOHNSON DOUGLAS WEBB,LANDER PETER AMBROSE,LOHMAN MARK CHRISTOPHER,PATEL VINOD FRANCIS,VEPACHEDU SREENIVASARAO,XIE YONGPING
- Priority: US15817599 1999-10-07; US16978499 1999-12-09
- Main IPC: A61P35/00
- IPC: A61P35/00 ; C07D471/04 ; C07D498/04 ; A61K31/4741 ; A61K31/4745
Abstract:
The present invention relates to a compound of formula (I), which are useful for inhibiting resistant neoplasms where the resistance is conferred in part or in total by MRP1.
Information query
IPC分类:
A | 人类生活必需 |
A61 | 医学或兽医学;卫生学 |
A61P | 化合物或药物制剂的特定治疗活性 |
A61P35/00 | 抗肿瘤药 |