Invention Application
- Patent Title: VITAMIN D RECEPTOR MODULATORS
- Patent Title (中): 维生素D受体调节剂
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Application No.: PCT/US2004/037182Application Date: 2004-11-16
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Publication No.: WO2005051893A2Publication Date: 2005-06-09
- Inventor: BUNEL, Emilio, Enrique , GAJEWSKI, Robert, Peter , JONES, Charles, David , LU, Jianliang , NAGPAL, Sunil , MA, Tianwei , YEE, Ying, Kwong
- Applicant: ELI LILLY AND COMPANY , BUNEL, Emilio, Enrique , GAJEWSKI, Robert, Peter , JONES, Charles, David , LU, Jianliang , NAGPAL, Sunil , MA, Tianwei , YEE, Ying, Kwong
- Applicant Address: Lilly Corporate Center, Indianapolis, IN 46285 US
- Assignee: ELI LILLY AND COMPANY,BUNEL, Emilio, Enrique,GAJEWSKI, Robert, Peter,JONES, Charles, David,LU, Jianliang,NAGPAL, Sunil,MA, Tianwei,YEE, Ying, Kwong
- Current Assignee: ELI LILLY AND COMPANY,BUNEL, Emilio, Enrique,GAJEWSKI, Robert, Peter,JONES, Charles, David,LU, Jianliang,NAGPAL, Sunil,MA, Tianwei,YEE, Ying, Kwong
- Current Assignee Address: Lilly Corporate Center, Indianapolis, IN 46285 US
- Agency: BOUDREAUX, William, R.
- Priority: US60/523,301 20031120
- Main IPC: C07C235/00
- IPC: C07C235/00
Abstract:
The present invention relates to novel, non-secosteroidal, hydroxyl substituted, carbon- linked diaryl compounds with vitamin D receptor (VDR) modulating activity that are less hypercalcemic than 1?,25 dihydroxy vitamin D3. These compounds are useful for treating bone disease and psoriasis.
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