Invention Application
WO2011039130A1 NEW BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS FXR AGONISTS
审中-公开
新的苯并咪唑衍生物及其作为FXR AGONISTS的用途
- Patent Title: NEW BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS FXR AGONISTS
- Patent Title (中): 新的苯并咪唑衍生物及其作为FXR AGONISTS的用途
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Application No.: PCT/EP2010/064217Application Date: 2010-09-27
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Publication No.: WO2011039130A1Publication Date: 2011-04-07
- Inventor: BENSON, Gregory Martin , BLEICHER, Konrad , FENG, Song , GRETHER, Uwe , KUHN, Bernd , MARTIN, Rainer E. , PLANCHER, Jean-Marc , RICHTER, Hans , RUDOLPH, Markus , TAYLOR, Sven
- Applicant: F. HOFFMANN-LA ROCHE AG , BENSON, Gregory Martin , BLEICHER, Konrad , FENG, Song , GRETHER, Uwe , KUHN, Bernd , MARTIN, Rainer E. , PLANCHER, Jean-Marc , RICHTER, Hans , RUDOLPH, Markus , TAYLOR, Sven
- Applicant Address: Grenzacherstrasse 124 CH-4070 Basel CH
- Assignee: F. HOFFMANN-LA ROCHE AG,BENSON, Gregory Martin,BLEICHER, Konrad,FENG, Song,GRETHER, Uwe,KUHN, Bernd,MARTIN, Rainer E.,PLANCHER, Jean-Marc,RICHTER, Hans,RUDOLPH, Markus,TAYLOR, Sven
- Current Assignee: F. HOFFMANN-LA ROCHE AG,BENSON, Gregory Martin,BLEICHER, Konrad,FENG, Song,GRETHER, Uwe,KUHN, Bernd,MARTIN, Rainer E.,PLANCHER, Jean-Marc,RICHTER, Hans,RUDOLPH, Markus,TAYLOR, Sven
- Current Assignee Address: Grenzacherstrasse 124 CH-4070 Basel CH
- Agency: WASCHBUESCH, Klaus
- Priority: EP09171700.9 20090929
- Main IPC: C07D235/18
- IPC: C07D235/18 ; C07D401/04 ; C07D403/10 ; C07D403/12 ; C07D405/14 ; C07D417/14 ; A61K31/4184 ; A61K31/4439
Abstract:
Compounds of formula (I) as well as pharmaceutically acceptable salts thereof can be used in the form of pharmaceutical compositions, wherein A, B, R 1 , R 2 , R 3 , R 4 , R 5 , n, m and p have the significance given in claim 1.
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