Invention Application
WO2012019428A8 BENZOHYDROL DERIVATIVES, A PREPARATION PROCESS AND PHARMACEUTICAL USE THEREOF
审中-公开
苯并呋喃衍生物,其制备方法和其药物用途
- Patent Title: BENZOHYDROL DERIVATIVES, A PREPARATION PROCESS AND PHARMACEUTICAL USE THEREOF
- Patent Title (中): 苯并呋喃衍生物,其制备方法和其药物用途
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Application No.: PCT/CN2011001252Application Date: 2011-08-01
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Publication No.: WO2012019428A8Publication Date: 2012-05-10
- Inventor: TANG PENGCHO , WU QINGQUAN , WU XIAO , ZHENG ZHEN , JI WENHAO
- Applicant: SHANGHAI HENGRUI PHARM CO LTD , JIANGSU HENGRUI MEDICINE CO , TANG PENGCHO , WU QINGQUAN , WU XIAO , ZHENG ZHEN , JI WENHAO
- Assignee: SHANGHAI HENGRUI PHARM CO LTD,JIANGSU HENGRUI MEDICINE CO,TANG PENGCHO,WU QINGQUAN,WU XIAO,ZHENG ZHEN,JI WENHAO
- Current Assignee: SHANGHAI HENGRUI PHARM CO LTD,JIANGSU HENGRUI MEDICINE CO,TANG PENGCHO,WU QINGQUAN,WU XIAO,ZHENG ZHEN,JI WENHAO
- Priority: CN201110112168 2011-04-25; CN201010249629 2010-08-10
- Main IPC: C07C271/16
- IPC: C07C271/16 ; A61K31/27 ; A61K31/343 ; A61K31/351 ; A61K31/353 ; A61P1/16 ; A61P3/10 ; A61P9/00 ; A61P9/04 ; A61P9/10 ; A61P9/12 ; A61P13/12 ; A61P25/00 ; A61P25/22 ; A61P25/28 ; A61P27/02 ; A61P43/00 ; C07D307/79 ; C07D309/04 ; C07D311/58 ; C07D407/12
Abstract:
Benzohydrol derivatives of formula (I), a preparation method, pharmaceutical compositions and pharmaceutical use thereof are disclosed in the invention. The derivatives can be used as rennin inhibitors to prepare the drugs for the treatment of the diseases related with rennin, such as antihypertensive drugs.
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