发明申请
WO2015056164A1 1,4-CYCLOHEXYLAMINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF
审中-公开
1,4-环己基胺衍生物及其制备方法
- 专利标题: 1,4-CYCLOHEXYLAMINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF
- 专利标题(中): 1,4-环己基胺衍生物及其制备方法
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申请号: PCT/IB2014/065293申请日: 2014-10-14
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公开(公告)号: WO2015056164A1公开(公告)日: 2015-04-23
- 发明人: TADDEI, Maurizio , CINI, Elena , RASPARINI, Marcello
- 申请人: CHEMO RESEARCH, S.L.
- 申请人地址: Quintanapalla 2 4ª planta E-28050 Madrid ES
- 专利权人: CHEMO RESEARCH, S.L.
- 当前专利权人: CHEMO RESEARCH, S.L.
- 当前专利权人地址: Quintanapalla 2 4ª planta E-28050 Madrid ES
- 代理机构: PALLADINO, Saverio Massimo et al.
- 优先权: ITMI2013A001693 20131014
- 主分类号: C07D233/61
- IPC分类号: C07D233/61 ; C07C275/26 ; C07D295/033 ; C07D295/04 ; C07D295/135
摘要:
The invention relates to a process for the synthesis of Cariprazine, an antipsychotic compound useful in the treatment of positive and negative symptoms associated to schizophrenia, with the following structural formula: (A) The invention further relates to the synthesis of intermediates useful in the preparation of Cariprazine.