公开(公告)号：EP2252606A1

公开(公告)日：2010-11-24

申请号：EP09710509.2

申请日：2009-02-10

Applicant: BASF SE

Inventor： LOHMANN, Jan Klaas ,  GLÄTTLI, Alice ,  GRAMMENOS, Wassilios ,  MONTAG, Jurith ,  MÜLLER, Bernd ,  VRETTOU, Marianna ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  RACK, Michael ,  DIETZ, Jochen

IPC: C07D401/12 ,  C07D403/12 ,  C07D413/12 ,  C07D417/12

CPC classification number: C07D401/12 ,  C07D401/14 ,  C07D403/12 ,  C07D413/12 ,  C07D417/12

Abstract: The present invention relates to pyrimidin-4-ylmethyl-sulfonamides of formula (I) wherein Ra, n, R, A, Y and Het are as defined in the claims and to the N-oxides, and salts thereof and their use for combating harmful fungi, and also to compositions and seed comprising at least one such compound. The invention also relates to a process for preparing these compounds.

Abstract translation: 本发明涉及式（I）的嘧啶-4-基甲基 - 磺酰胺，其中Ra，n，R，A，Y和Het如权利要求中所定义，并且涉及N-氧化物及其盐以及它们用于防治 有害真菌，并且还涉及包含至少一种这样的化合物的组合物和种子。 本发明还涉及制备这些化合物的方法。

公开(公告)号：EP2231605A1

公开(公告)日：2010-09-29

申请号：EP08857320.9

申请日：2008-11-21

Applicant: BASF SE

Inventor： GRAMMENOS, Wassilios ,  LOHMANN, Jan Klaas ,  GROTE, Thomas ,  DIETZ, Jochen ,  MÜLLER, Bernd ,  PUHL, Michael ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  VRETTOU, Marianna ,  RHEINHEIMER, Joachim

IPC: C07D213/71 ,  C07D213/74 ,  C07D401/12 ,  C07D413/12 ,  C07D417/12 ,  C07D213/643 ,  C07D213/30 ,  C07D213/69 ,  C07D213/70 ,  C07D213/79 ,  C07D217/24 ,  C07D237/14 ,  C07D237/16 ,  C07D239/34 ,  C07D239/54

CPC classification number: C07D213/643 ,  A01N43/40 ,  A01N43/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/78 ,  A01N43/80 ,  C07D213/30 ,  C07D213/69 ,  C07D213/70 ,  C07D213/71 ,  C07D213/74 ,  C07D213/79 ,  C07D217/24 ,  C07D237/14 ,  C07D237/16 ,  C07D239/34 ,  C07D239/54 ,  C07D239/60 ,  C07D261/08 ,  C07D261/12 ,  C07D277/24 ,  C07D277/34 ,  C07D401/12 ,  C07D413/12 ,  C07D417/12 ,  A01N37/34 ,  A01N43/653 ,  A01N47/04 ,  A01N47/24 ,  A01N2300/00

Abstract: The present invention relates to novel pyridylmethyl-sulfonamide compounds of formula (I) where: n is 0 to 4; m is 0 to 4; R1 is halogen, CN, NO2, OH, SH, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, etc.; and/or two radicals R1 together form a fused ring; R2 is H, C1-C4-alkyl, C1-C4-haloalkyl, C2-C4-alkenyl, C2-C4-alkynyl, C3-C8-cycloalkyl, C1-C4-alkyl-C3-C8-cycloalkyl or benzyl; R3 is halogen, CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy; Y is -O-, C1-C4-alkane- diyl, -O-CH2-, -CH2-O-, -C(NOR')-, -S-, -S(=0)-, -Sf=O)2- or -N(R')-; and the N-oxides, and salts thereof and their use for combating phytopathogenic harmful fungi, and also to compositions and seed comprising at least one such compound.

公开(公告)号：EP2117312A1

公开(公告)日：2009-11-18

申请号：EP08701270.4

申请日：2008-01-07

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  GRAMMENOS, Wassilios ,  MÜLLER, Bernd ,  LOHMANN, Jan, Klaas ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  VRETTOU, Marianna

IPC: A01N43/90 ,  C07D487/04 ,  A01P3/00

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: Azolopyrimidines of the formula (I), wherein the symbols have the meanings provided in the description, are suited to fight plant pathogenic fungi.

公开(公告)号：EP1504001B1

公开(公告)日：2009-04-15

申请号：EP03742510.5

申请日：2003-02-06

Applicant: BASF SE

Inventor： SCHIEWECK, Frank ,  TORMO I BLASCO, Jordi ,  GROTE, Thomas ,  GYPSER, Andreas ,  MÜLLER, Bernd ,  RHEINHEIMER, Joachim ,  ROSE, Ingo ,  SCHÄFER, Peter ,  GRAMMENOS, Wassilios ,  GEWEHR, Markus ,  SCHWÖGLER, Anja ,  BLETTNER, Carsten ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried ,  LORENZ, Gisela ,  STIERL, Reinhard

IPC: C07D401/04 ,  A01N43/54

CPC classification number: C07D401/04

Abstract: The invention relates to 2-(2-pyridyl)-5-phenyl-6-aminopyrimidines of formula I, wherein the substitutes and the index have the following meaning: R1 represents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino, dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m = 0 or 1 - 4; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3, R4 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, R3 and R4 together with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; R5 represents halogen, alkyl or halogenalkyl; R6 represents hydrogen or one of the known groups in R5; R7, R8 represent hydrogen, halogen, alkyl or halogenalkyl; R9 represents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants.

公开(公告)号：EP2010515A1

公开(公告)日：2009-01-07

申请号：EP07727984.2

申请日：2007-04-11

Applicant: BASF SE

Inventor： GRAMMENOS, Wassilios ,  GROTE, Thomas ,  DIETZ, Jochen ,  LOHMANN, Jan, Klaas ,  RENNER, Jens ,  MÜLLER, Bernd ,  ULMSCHNEIDER, Sarah

IPC: C07D401/04 ,  C07D401/14 ,  C07D405/14 ,  C07D409/14 ,  C07D491/048 ,  C07D491/052 ,  C07D491/056 ,  A01N43/54 ,  A01N43/90

CPC classification number: C07D401/04 ,  A01N43/54 ,  A01N43/90 ,  C07D401/14 ,  C07D405/14 ,  C07D409/14 ,  C07D491/04

Abstract: The invention relates to 2-(pyridin-2-yl)-pyrimidines of formula (I) and their use in the control of parasitic fungi and to herbicides that contain said compounds as an effective ingredient thereof. In formula (I), Q represents a condensed, saturated five-, six- or seven-membered carbocycle or five-, six- or seven-membered heterocycle which, in addition to the carbon ring members, has one or two heteroatoms selected from oxygen and sulfur as the ring members, the carbocycle and the heterocycle being unsubstituted or having 1, 2, 3 or 4 C1-C4 alkyl groups as the substituents; R1 represents hydrogen, OH, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy or halogen; R2 represents hydrogen, NO2, halogen, C1-C6 alkyl, C3-C6 cycloalkyl, C1-C6 alkoxy, C1-C6 halogenalkyl or C1-C6 halogenalkoxy; R3 represents hydrogen, halogen, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl or C1-C4 halogenalkoxy; R4 has phenyl, 5-membered heteroaryl which has 1, 2, 3 or 4 nitrogen atoms or 1 heteroatom selected from oxygen and sulfur and optionally 1, 2 or 3 nitrogen atoms as the ring atoms, or 6-membered hetaryl, which has 1, 2, 3 or 4 nitrogen atoms as the ring members, wherein phenyl, 5- and 6-membered hetaryl may have 1, 2, 3 or 4 substituents Ra.

公开(公告)号：EP1909580A1

公开(公告)日：2008-04-16

申请号：EP06792534.7

申请日：2006-07-20

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  GROTE, Thomas ,  HÜNGER, Udo ,  LOHMANN, Jan Klaas ,  MÜLLER, Bernd ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  GRAMMENOS, Wassilios ,  RHEINHEIMER, Joachim

IPC: A01N43/90 ,  C07D487/04

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to 5-methyl-6-phenyl-triazolopyrimidinyl amines of formula (I) wherein the substituents have the designations cited in the description. The invention also relates to methods for producing said compounds, to agents containing the same, and to the use thereof for controlling plant pathogenic fungi.

Abstract translation: 本发明涉及式（I）的5-甲基-6-苯基 - 三唑并嘧啶胺，其中取代基具有在说明书中引用的名称。 本发明还涉及生产所述化合物的方法，含有所述化合物的试剂，以及其用于防治植物病原真菌的用途。

公开(公告)号：EP1697365B1

公开(公告)日：2008-03-05

申请号：EP04803851.7

申请日：2004-12-14

Applicant: BASF SE

Inventor： TORMO I BLASCO, Jordi ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  STIERL, Reinhard

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to 6-(2-halogen-4-alcoxyphenyl)-triazolopyrimidine of formula (I), wherein substituents have the following significance: R1 is alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalcenyl, cycloalkenyl, halogenocycloalkenyl, alkynyl, halogenoalkynyl, cycloalkynyl, halogencycloalkynyl or phenyl, naphthyl or a type of heterocycle having from 5 to 6 saturated, partially saturated or aromatic chains containing one or four heteroatoms of a O, N and S group; R2 is hydrogen or one of groups mentioned in R1, R1 and R2 can also form together with a nitrogen atom to which they are linked a 5 or 6-links heterocycle or a heteroaryl which is linked by N and can contain from one to three other heteroatoms of the O, N and S group in the form of a ring link; R3 is alkyl, halogenalkyl, alcenyl, halogenalcenyl, alcynyl, halogenoalkynyl, phenylalkyl, mono or dialcoxyalkyl; R1, R2 and/or R3 can be substituted according to a description; L is hydrogen, fluoride or chlorine; x is cyano, alkyl, alkoxy, alkenyloxy, halogenalkoxy or halogenalkenyloxy;. A method for producing said compounds, the agents containing said compounds and the use thereof against phytopathogenic harmful fungus are also disclosed.

公开(公告)号：EP2935236B1

公开(公告)日：2017-11-29

申请号：EP13810923.6

申请日：2013-12-12

Applicant: BASF SE

Inventor： GRAMMENOS, Wassilios ,  CRAIG, Ian Robert ,  BOUDET, Nadege ,  MÜLLER, Bernd ,  DIETZ, Jochen ,  LAUTERWASSER, Erica May Wilson ,  LOHMANN, Jan Klaas ,  GROTE, Thomas ,  HADEN, Egon ,  ESCRIBANO CUESTA, Ana

IPC: C07D401/04 ,  C07D401/06 ,  C07D401/12 ,  C07D403/04 ,  C07D403/06 ,  C07D403/12 ,  C07D417/04 ,  C07D417/06 ,  C07D417/12 ,  A01N43/50 ,  A01N43/54 ,  A01N43/653 ,  A01N43/78

CPC classification number: C07D249/08 ,  A01N43/653 ,  A01N43/78 ,  A01N43/82 ,  C07D401/04 ,  C07D401/06 ,  C07D401/10 ,  C07D401/12 ,  C07D403/04 ,  C07D403/06 ,  C07D403/12 ,  C07D409/10 ,  C07D417/04 ,  C07D417/06 ,  C07D417/10 ,  C07D417/12

公开(公告)号：EP2744790B1

公开(公告)日：2016-04-27

申请号：EP12745877.6

申请日：2012-08-14

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  RIGGS, Richard ,  BOUDET, Nadege ,  LOHMANN, Jan Klaas ,  CRAIG, Ian Robert ,  HADEN, Egon ,  LAUTERWASSER, Erica May Wilson ,  MÜLLER, Bernd ,  GRAMMENOS, Wassilios ,  GROTE, Thomas

IPC: C07D249/08 ,  A01N43/653

CPC classification number: A01N43/653 ,  C07D249/08

公开(公告)号：EP2952507A1

公开(公告)日：2015-12-09

申请号：EP14171469.1

申请日：2014-06-06

Applicant: BASF SE

Inventor： GRAMMENOS, Wassilios ,  BOUDET, Nadege ,  MÜLLER, Bernd ,  QUINTERO PALOMAR, Maria Angelica ,  ESCRIBANO CUESTA, Ana ,  LAUTERWASSER, Erica May Wilson ,  LOHMANN, Jan Klaas ,  GROTE, Thomas ,  KRETSCHMER, Manuel ,  CRAIG, Ian Robert

IPC: C07D249/08 ,  A01N43/653

CPC classification number: C07D249/08 ,  A01N43/653

Abstract: The present invention relates to compounds of the formula I

wherein the variables are defined in the description and claims, their preparation and uses thereof.

Abstract translation: 本发明涉及式I化合物，其中变量在说明书和权利要求书中定义，其制备和用途。