公开(公告)号：EP1504001B1

公开(公告)日：2009-04-15

申请号：EP03742510.5

申请日：2003-02-06

Applicant: BASF SE

Inventor： SCHIEWECK, Frank ,  TORMO I BLASCO, Jordi ,  GROTE, Thomas ,  GYPSER, Andreas ,  MÜLLER, Bernd ,  RHEINHEIMER, Joachim ,  ROSE, Ingo ,  SCHÄFER, Peter ,  GRAMMENOS, Wassilios ,  GEWEHR, Markus ,  SCHWÖGLER, Anja ,  BLETTNER, Carsten ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried ,  LORENZ, Gisela ,  STIERL, Reinhard

IPC: C07D401/04 ,  A01N43/54

CPC classification number: C07D401/04

Abstract: The invention relates to 2-(2-pyridyl)-5-phenyl-6-aminopyrimidines of formula I, wherein the substitutes and the index have the following meaning: R1 represents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino, dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m = 0 or 1 - 4; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3, R4 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, R3 and R4 together with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; R5 represents halogen, alkyl or halogenalkyl; R6 represents hydrogen or one of the known groups in R5; R7, R8 represent hydrogen, halogen, alkyl or halogenalkyl; R9 represents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants.

公开(公告)号：EP1697365B1

公开(公告)日：2008-03-05

申请号：EP04803851.7

申请日：2004-12-14

Applicant: BASF SE

Inventor： TORMO I BLASCO, Jordi ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  STIERL, Reinhard

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to 6-(2-halogen-4-alcoxyphenyl)-triazolopyrimidine of formula (I), wherein substituents have the following significance: R1 is alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalcenyl, cycloalkenyl, halogenocycloalkenyl, alkynyl, halogenoalkynyl, cycloalkynyl, halogencycloalkynyl or phenyl, naphthyl or a type of heterocycle having from 5 to 6 saturated, partially saturated or aromatic chains containing one or four heteroatoms of a O, N and S group; R2 is hydrogen or one of groups mentioned in R1, R1 and R2 can also form together with a nitrogen atom to which they are linked a 5 or 6-links heterocycle or a heteroaryl which is linked by N and can contain from one to three other heteroatoms of the O, N and S group in the form of a ring link; R3 is alkyl, halogenalkyl, alcenyl, halogenalcenyl, alcynyl, halogenoalkynyl, phenylalkyl, mono or dialcoxyalkyl; R1, R2 and/or R3 can be substituted according to a description; L is hydrogen, fluoride or chlorine; x is cyano, alkyl, alkoxy, alkenyloxy, halogenalkoxy or halogenalkenyloxy;. A method for producing said compounds, the agents containing said compounds and the use thereof against phytopathogenic harmful fungus are also disclosed.

公开(公告)号：EP1856055B1

公开(公告)日：2014-10-01

申请号：EP06708289.1

申请日：2006-02-15

Applicant: BASF SE

Inventor： GEWEHR, Markus ,  DIETZ, Jochen ,  GROTE, Thomas ,  BLETTNER, Carsten ,  GRAMMENOS, Wassilios ,  HÜNGER, Udo ,  MÜLLER, Bernd ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  LOHMANN, Jan Klaas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  STRATHMANN, Siegfried ,  STIERL, Reinhard

IPC: C07D231/14 ,  A01N43/56

CPC classification number: C07D231/14 ,  A01N43/56

公开(公告)号：EP1725560B1

公开(公告)日：2010-07-07

申请号：EP05715825.5

申请日：2005-03-08

Applicant: BASF SE

Inventor： TORMO I BLASCO, Jordi ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  NIEDENBRÜCK, Matthias ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  STIERL, Reinhard

IPC: C07D487/04 ,  A01N43/90

CPC classification number: C07D487/04

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, alkoxymethylene or alkoxyethylene, whereby the aliphatic groups can be substituted according to the description and R2 represents n-propyl or n-butyl. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

公开(公告)号：EP2550666A2

公开(公告)日：2013-01-30

申请号：EP11758892.1

申请日：2011-03-17

Applicant: BASF SE

Inventor： BLETTNER, Carsten ,  KACZUN, Jürgen ,  KRESS, Ria ,  WIEBELHAUS, Dag

IPC: H01F1/047 ,  B22F1/00

CPC classification number: H01F41/0266 ,  B29C43/003 ,  H01F1/0558 ,  H01F1/0578 ,  H01F1/26 ,  H01F41/0246

Abstract: The invention relates to a composition for producing magnetic or magnetizable moldings, comprising from 95.5 to 98.95% by weight of a powder made of a magnetic or magnetizable material, from 1.0 to 4% by weight of a mixture made of at least one epoxy-novolak resin, and also of at least one hardener, and comprising from 0.05 to 0.5% by weight of at least one additive, based in each case on the total weight of the composition. The mixture made of the at least one epoxy-novolak resin and of the at least one hardener comprises from 85 to 95% by weight of the epoxy-novolak resin and from 5 to 15% by weight of hardener. The hardener has been selected from (cyclo)aliphatic amines and their adducts, polyamides, Mannich bases, amidoamines, phenolic resins, imidazoles, and imidazole derivatives, dicyandiamide, and BF3-monoethanolamine. The invention further relates to a process for producing the composition, and also to a process for producing a molding made of the composition.

公开(公告)号：EP1761499B1

公开(公告)日：2010-02-24

申请号：EP05759346.9

申请日：2005-06-11

Applicant: BASF SE

Inventor： GEWEHR, Markus ,  MÜLLER, Bernd ,  GROTE, Thomas ,  GRAMMENOS, Wassilios ,  SCHWÖGLER, Anja ,  RHEINHEIMER, Joachim ,  BLETTNER, Carsten ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  WAGNER, Oliver ,  WERNER, Frank ,  RETHER, Jan ,  STRATHMANN, Siegfried ,  STIERL, Reinhard ,  SCHERER, Maria

IPC: C07D231/14 ,  A01N43/56

CPC classification number: C07D231/14

Abstract: The invention relates to 1-methyl-3-trifluoromethyl-pyrazole-4-carboxylic acid-(ortho-phenyl)-anilides of formula I, wherein the substituents have the following meaning: R1 and R 2 independently represent halogen, C1-C6-alkyl, C1-C6 halogen-alkyl, cyano, nitro, methoxy, trifluoromethoxy or difluoromethoxy; under the proviso that if R2 represents chlorine in the 4-position, R1 does not represent trifluoromethyl in the 3 position.

公开(公告)号：EP1725561B1

公开(公告)日：2010-07-07

申请号：EP05715826.3

申请日：2005-03-08

Applicant: BASF SE

Inventor： TORMO I BLASCO, Jordi ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  NIEDENBRÜCK, Matthias ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  STIERL, Reinhard

IPC: C07D487/04 ,  A01N43/90

CPC classification number: C07D487/04

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl or alkoxyalkyl, whereby the aliphatic groups can be substituted according to the description; R2 represents CHR3CH3, cyclopropyl, CH=CH2 or CH2CH=CH2 and R3 represents hydrogen, CH3 or CH2CH3. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

公开(公告)号：EP2172466A1

公开(公告)日：2010-04-07

申请号：EP09179928.8

申请日：2005-07-22

Applicant: BASF SE

Inventor： GRAMMENOS, Wassilios ,  GROTE, Thomas ,  BLETTNER, Carsten ,  GEWEHR, Markus ,  HÜNGER, Udo ,  MÜLLER, Bernd ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  SCHÖFL, Ulrich ,  KÖHLE, Harald ,  STRATHMANN, Siegfried ,  SCHERER, Maria ,  STIERL, Reinhard ,  RETHER, Jan

IPC: C07D401/04 ,  A01N43/54

CPC classification number: C07D401/04

Abstract: Die vorliegende Erfindung betrifft 2-(Pyridin -2-yl)-pyrimidine Verbindungen der allgemeinen Formel I und ihre Verwendung zur Bekämpfung von Schadpilzen sowie Pflanzenschutzmittel, die derartige Verbindungen als wirksamen Bestandteil enthalten.

Hierin steht k für 0, 1, 2 oder 3, m für 0, 1, 2, 3, 4 oder 5, n für 1, 2, 3, 4 oder 5;
R 1 bedeuten unabhängig voneinander Halogen, OH, CN, NO 2 C 1 -C 4 -Alkyl, C 1 -C 4 -Halogenalkyl, C 1 -C 4 -Alkoxy, C 1 -C 4 -Halogenalkoxy, C 2 -C 4 -Alkenyl, C 2 -C 4 -Alkinyl, C 3 -C 8 -Cycloalkyl, C 1 -C 4 -Alkoxy-C 1 -C 4 -alkyl, Amino, Phenoxy, das gegebenenfalls durch Halogen oder C 1 -C 4 -Alkyl substituiert ist, NHR, NR 2 , C(R a )=N-OR b , S(=O) p A 1 oder C(=O)A 2 , oder zwei an benachbarte C-Atome gebundene Reste R 1 können auch gemeinsam für eine Gruppe -O-Alk-O- stehen, worin Alk für lineares oder verzweigtes C 1 -C 4 -Alkylen steht, worin 1, 2, 3 oder 4 Wasserstoffatome auch durch Halogen ersetzt sein können;
R 2 C 1 -C 4 -Halogenalkyl, C 1 -C 4 -Alkoxy, C 1 -C 4 -Halogenalkoxy, Hydroxy, Halogen, CN oder NO 2 bedeutet; wobei R 2 auch Wasserstoff oder C 1 -C 4 -Alkyl bedeuten kann, wenn wenigstens eine der drei folgenden Bedingungen erfüllt ist:
- n steht für 3, 4 oder 5,
- k steht für 1, 2 oder 3,
- für m ≠ 0 steht wenigstens einer der Reste R 1 für einen von Halogen, C 1 -C 4 -Alkyl, C 1 -C 4 -Alkoxy und C 1 -C 4 -Halogenalkyl verschieden Rest; und
R 3 für C 1 -C 4 -Alkyl.

Abstract translation: 2-吡啶基嘧啶衍生物（I）是新的。 式（I）的2-吡啶基嘧啶衍生物及其盐是新的。 k：0-3; m：0-5; n：1-5; R 1>卤素，OH，CN，NO 2，1-4C（卤素）烷基，104C（卤素）烷氧基，2-4C烯基，2-4C炔基，3-8C环烷基，（1-4C）烷氧基（1- 4C）烷基，NH 2，苯氧基（任选被卤素或1-4C烷基取代），NHR，NRR，C（Ra）= NORb，SO pA 1>或COA 2>; 或R 1> R 1→1-4C（卤代）亚烷基二氧基; R：1-4C烷基或1-4C烷基羰基; Ra：H或1-4C烷基; Rb：1-4C烷基，3-4C烯基或3-4C炔基; p：0-2; 当p = 2时，1→1-4C烷基或NH 2，1-4C烷基氨基或二（1-4C烷基）氨基; A 2 H，OH，1-4C烷基，1-4C烷基氨基，二（1-4C烷基）氨基，2-4C烯基或1-4C（卤代）烷氧基; R 2> 1-4C卤代烷基，1-4C（卤代）烷氧基，OH，卤素，CN或NO 2，或R 2可以是H或1-4C烷基，如果n = 3-5和/或k = 1- 3和/或至少一个R 1>不是卤素，1-4C（卤代）烷基和1-4C烷氧基; 和R 3> 1-4C烷基。 还包括通过用化合物（I）处理待保护免受真菌侵袭的真菌或材料，植物，土壤或种子进行真菌侵袭来控制植物病原性真菌的独立权利要求。 活动：植物抗真菌。 在对番茄植物上的链格孢（Alternaria solani）的保护性试验中，用2-（5-甲基-6-苯基-2-吡啶基）-4,5-五亚甲基 - 嘧啶（250ppm）处理的植物没有受到攻击，而90％ 植物受到攻击。 行动机制：无给予。

公开(公告)号：EP1773806B1

公开(公告)日：2010-02-24

申请号：EP05761662.5

申请日：2005-07-22

Applicant: BASF SE

Inventor： GRAMMENOS, Wassilios ,  GROTE, Thomas ,  BLETTNER, Carsten ,  GEWEHR, Markus ,  HÜNGER, Udo ,  MÜLLER, Bernd ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  SCHÖFL, Ulrich ,  KÖHLE, Harald ,  STRATHMANN, Siegfried ,  SCHERER, Maria ,  STIERL, Reinhard ,  RETHER, Jan

IPC: C07D401/04 ,  A01N43/54

CPC classification number: C07D401/04

Abstract: The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type, whereby: k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)=N-ORb, S(=O)pA1 or C(=O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group -O-Alk-O-, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

公开(公告)号：EP1663976B1

公开(公告)日：2009-12-30

申请号：EP04765053.6

申请日：2004-09-10

Applicant: BASF SE

Inventor： GRAMMENOS, Wassilios ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  TORMO I BLASCO, Jordi ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  GÖTZ, Norbert ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  SCHERER, Maria ,  STIERL, Reinhard

IPC: C07D213/42

CPC classification number: C04B35/632 ,  C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12

Abstract: The invention relates to sulphonamides of formula (I) in which the substituents have the following meanings: R1 = H, alkyl, alkoxy, alkenyl or alkinyl and R2, R3, R4, R5 = hydrogen, halogen, alkyl, alkoxy or halomethyl; R2 and R3 can also together form a phenyl, cyclopentyl, or cyclohexyl ring, whereby said ring can carry R2' and R3', where R2', R3' = H, halogen, alkyl, alkoxy or halomethyl; in the case a), when R2, R3, R4 and R5 = H, X = phenyl, substituted with a group -C(R6)=NOR7, where R6= alkyl and R7 = alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkinyl or haloalkinyl and in case b), when at least one of the groups R2, R3, R4 and R5 is not H, X = phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated, or aromatic heterocycle, bonded by means of a C atom, comprising one to four heteroatoms from the group O, N or S, where X can be substituted as per the description. The invention further relates to methods for production of said compounds, agents comprising the same and use thereof for the control of fungal pests which are pathogenic to plants.