公开(公告)号：EP1751162A1

公开(公告)日：2007-02-14

申请号：EP05744598.3

申请日：2005-05-13

申请人： BASF Aktiengesellschaft

发明人： BLETTNER, Carsten ,  SCHIEWECK, Frank ,  TORMO, I. Blasco, Jordi ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  SPEAKMAN, John-Bryan ,  Jabs, Thorsten ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  SCHERER, Maria ,  STIERL, Reinhard

IPC分类号： C07D487/04 ,  A01N43/90

CPC分类号： A01N43/90 ,  C07D487/04

摘要： The invention relates to novel triazolopyrimidine compounds of general formula (I), to their use for controlling pathogenic fungi and to agricultural pesticides containing compounds of this type as active constituents. In formula (I), X, Y, L, m, Ar and A are defined as follows: X represents halogen, cyano, C1-C4 alkyl, C1-C4 haloalkyl, C1-C4 alkoxy or C1-C4 haloalkoxy; Y represents halogen, C1-C4 alkyl or C1-C4 haloalkyl; L represents independently of one another halogen, C1-C6 alkyl, C2-C6 alkenyl, C1-C6 haloalkyl, C1-C6 alkoxy, C1-C6 haloalkoxy, nitro, amino, NHR, NR2, cyano, S(=O)nA1 or C(=O)A2; m represents 0, 1, 2, 3 or 4; A stands for a chemical bond or a CR4R5 group; Ar represents phenyl or a 5- or 6-membered heteroaromatic group comprising 1, 2 or 3 heteroatoms selected from O, S and N as ring members, whereby the phenyl and the heteroaromatic group can comprise a fused benzole ring and can have 1, 2, 3, 4 or 5 Ra substituents. R1 to R3 are defined as cited in claim 1.

摘要翻译： 本发明涉及通式（I）的新三唑并嘧啶化合物，它们用于防治病原真菌的用途以及含有这类化合物作为活性成分的农用杀虫剂。 在式（I）中，X，Y，L，m，Ar和A定义如下：X代表卤素，氰基，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4烷氧基或C 1 -C 4卤代烷氧基; Y代表卤素，C 1 -C 4烷基或C 1 -C 4卤代烷基; L彼此独立地表示卤素，C 1 -C 6烷基，C 2 -C 6烯基，C 1 -C 6卤代烷基，C 1 -C 6烷氧基，C 1 -C 6卤代烷氧基，硝基，氨基，NHR，NR 2， C（= O）A2; m代表0,1,2,3或4; A代表化学键或CR4R5基团; Ar表示苯基或包含1,2或3个选自O，S和N的杂原子作为环成员的5或6元杂芳族基团，其中苯基和杂芳族基团可包含稠合的苯并环并且可具有1,2 ，3,4或5个Ra取代基。 R1至R3如权利要求1中所定义。

公开(公告)号：EP1751160A1

公开(公告)日：2007-02-14

申请号：EP04803834.3

申请日：2004-12-14

申请人： BASF Aktiengesellschaft

发明人： TORMO I BLASCO, Jordi ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  STIERL, Reinhard

IPC分类号： C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04

摘要： The invention relates to 6-(2,3,6-trifluorophenyl)-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R2 represents hydrogen or one of the groups cited for R1; R1 and R2, together with the nitrogen atom, to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded via N and can contain one to three additional heteroatoms from the groups O, N and S as a ring member; R1 and/or R2 can be substituted in accordance with the description; X represents cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy. The invention also relates to methods for producing said compounds, to agents containing the latter and to their use for combating plant-pathogenic fungi.

公开(公告)号：EP1746892A2

公开(公告)日：2007-01-31

申请号：EP05744652.8

申请日：2005-05-11

申请人： BASF Aktiengesellschaft

发明人： BLETTNER, Carsten ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  HÜNGER, Udo ,  MÜLLER, Bernd ,  NIEDENBRÜCK, Matthias ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  NAVE, Barbara ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  STIERL, Reinhard

IPC分类号： A01N43/90

CPC分类号： A01N43/90 ,  A01N59/06 ,  A01N59/02 ,  A01N57/12 ,  A01N47/38 ,  A01N47/34 ,  A01N47/24 ,  A01N47/04 ,  A01N43/50 ,  A01N43/76 ,  A01N43/653 ,  A01N43/36 ,  A01N43/40 ,  A01N43/32 ,  A01N37/48 ,  A01N37/46 ,  A01N37/38 ,  A01N37/34 ,  A01N2300/00

摘要： The invention relates to fungicidal mixtures containing in the form of active components 1) 5-methyl-7-amino-triazolopyrimidine of formula (I), wherein R1 is alkyl, halogenalkyl, alkenyl or cyclopentyl, R2 is hydrogen or alkyl, R1 and R2 together with the nitrogen atom to which they are bound may form a piperidinyl cycle substitutable by a methyl group, L1 is fluorine or chlorine, L2, L3 are independently from each other hydrogen, fluorine or chlorine and 2) at least one type of active substance selected from groups A) azoles, B) strobilurins, C) acyl alanines, D) amine derivatives, E) anilinopyrimidines; F) dicarboximides; G) cinnamic acid amides and analogues thereof, H) antibiotics, K) dithiocarbamates, L) heterocyclic compounds, M) sulphur and copper fungicides, N) nitrophenyl derivatives, O) phenylpyrroles, P) sulfenic acid derivatives, Q) other fungicides and R) growth retardants according to the descriptions, wherein said mixtures contain the compounds in a synergically efficient amount. Novel triazolopyrimidines, methods for controlling pathogenic fungi using the mixtures of the compound (I) with active substances of the groups A) and R), the use the compounds (I) with the active substances of the groups A) and R) for producing said mixtures and agents containing said mixtures are also disclosed.

公开(公告)号：EP1725557A1

公开(公告)日：2006-11-29

申请号：EP05700961.5

申请日：2005-01-15

申请人： BASF Aktiengesellschaft

发明人： TORMO I BLASCO, Jordi ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  STIERL, Reinhard

IPC分类号： C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to substituted triazolopyrimidines of formula (I), with the substituents as follows: R1, R2 = H, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkinyl, haloalkinyl, phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, comprising one to four heteroatoms of the group O, N or S, R1 and R2 can, together with the nitrogen atom to which it is attached, form a five- or six-membered heterocycle or heteroaryl, bonded via N and containing one to three further heteroatoms from the group O, N and S as ring members, substituted as per the description, L1 = fluorine, chlorine or bromine, L2 = H, alkyl or alkoxy and X = halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy. The invention further relates to methods and intermediates for production of said compounds, agents comprising the same and use thereof for controlling fungal pests harmful to plants.

公开(公告)号：EP1699752A1

公开(公告)日：2006-09-13

申请号：EP04804217.0

申请日：2004-12-22

申请人： BASF Aktiengesellschaft

发明人： GEWEHR, Markus ,  MÜLLER, Bernd ,  GROTE, Thomas ,  GRAMMENOS, Wassilios ,  TORMO I BLASCO, Jordi ,  SCHWÖGLER, Anja ,  RHEINHEIMER, Joachim ,  BLETTNER, Carsten ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  WAGNER, Oliver ,  SPEAKMAN, John-Bryan ,  RETHER, Jan ,  STRATHMANN, Siegfried ,  STIERL, Reinhard

IPC分类号： C07C251/38 ,  C07D213/82 ,  C07D207/34 ,  C07D263/34 ,  C07D277/56 ,  C07D279/12 ,  C07D307/30 ,  C07D307/54 ,  C07D307/71 ,  C07D333/38 ,  A01N43/10 ,  A01N43/40 ,  A01N43/56 ,  A01N43/74

CPC分类号： C07D213/82 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01N47/48 ,  C07C251/38 ,  C07D207/34 ,  C07D231/14 ,  C07D263/34 ,  C07D277/56 ,  C07D279/12 ,  C07D307/30 ,  C07D307/54 ,  C07D307/71 ,  C07D333/38

摘要： The invention relates to (hetero)cyclyl carboxanilides of general formula (I), wherein n represents 0, 1, 2, 3, or 4, m represents 1, 2, or 3, Y represents oxygen or sulfur, A represents optionally substituted phenyl or an at least monounsaturated, optionally substituted five-membered or six-membered heterocycle, and R1, R2, R3m, R4, R5, and R6 have the meanings indicated in claim 1, and the agriculturally useful salts thereof. The invention further relates to the use of said (hetero)cyclyl carboxanilides of general formula (I) and the agriculturally useful salts thereof as fungicides as well as plant protection agents containing the same.

公开(公告)号：EP1697367A1

公开(公告)日：2006-09-06

申请号：EP04803941.6

申请日：2004-12-16

申请人： BASF Aktiengesellschaft

发明人： TORMO I BLASCO, Jordi ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  STIERL, Reinhard

IPC分类号： C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to triazolopyrimidines of formula (I) in which the substituents are defined as follows: R1, R2 represent hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R1 and R2, together with the nitrogen atom, to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded via N, can contain an additional heteroatom from the group O, N and S as a ring member and can be substituted according to the description; L1, L2 represent hydrogen, cyano, haloalkyl, alkoxy, alkenyloxy or C(=O)A, whereby at least one group L1 or L2 does not represent hydrogen; A represents hydrogen, hydroxy, alkyl, alkoxy, haloalkoxy, C1-C8 alkylamino or dialkylamino; L3 represents hydrogen, halogen, cyano, nitro, haloalkyl, alkoxy or alkoxycarbonyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to their use for combating plant-pathogenic fungi.

公开(公告)号：EP1689750A1

公开(公告)日：2006-08-16

申请号：EP04797968.7

申请日：2004-11-18

申请人： BASF Aktiengesellschaft

发明人： TORMO I BLASCO, Jordi ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  STIERL, Reinhard

IPC分类号： C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04

摘要： Disclosed are 6-(2,4,6-trifluorophenyl)-triazolopyrimidines of formula (I), wherein the substituents have the following meaning: R1 represents alkyl, alkyl halide, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkinyl, haloalkinyl, or cycloalkinyl, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group comprising O, N, and S; R2 represents hydrogen or one of the groups mentioned for R1, R1 and R2 also optionally forming a five-membered or six-membered ring along with the nitrogen atom to which the same are bonded, said ring being interrupted by an atom from the group comprising O, N, and S, and/or R1 and/or R2 being optionally substituted according to the description; X represents cyano, C1-C4 alkoxy, C3-C4 alkenyloxy, C1-C2 haloalkoxy, or C3-C4 haloalkenyloxy. Also disclosed are a method for producing said compounds, substances containing the same, and the use thereof for controlling plant-pathogenic fungi.

公开(公告)号：EP1663976A1

公开(公告)日：2006-06-07

申请号：EP04765053.6

申请日：2004-09-10

申请人： BASF Aktiengesellschaft

发明人： GRAMMENOS, Wassilios ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  TORMO I BLASCO, Jordi ,  GROTE, Thomas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  GÖTZ, Norbert ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  SCHERER, Maria ,  STIERL, Reinhard

IPC分类号： C07D213/42

CPC分类号： C04B35/632 ,  C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12

摘要： The invention relates to sulphonamides of formula (I) in which the substituents have the following meanings: R1 = H, alkyl, alkoxy, alkenyl or alkinyl and R2, R3, R4, R5 = hydrogen, halogen, alkyl, alkoxy or halomethyl; R2 and R3 can also together form a phenyl, cyclopentyl, or cyclohexyl ring, whereby said ring can carry R2' and R3', where R2', R3' = H, halogen, alkyl, alkoxy or halomethyl; in the case a), when R2, R3, R4 and R5 = H, X = phenyl, substituted with a group -C(R6)=NOR7, where R6= alkyl and R7 = alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkinyl or haloalkinyl and in case b), when at least one of the groups R2, R3, R4 and R5 is not H, X = phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated, or aromatic heterocycle, bonded by means of a C atom, comprising one to four heteroatoms from the group O, N or S, where X can be substituted as per the description. The invention further relates to methods for production of said compounds, agents comprising the same and use thereof for the control of fungal pests which are pathogenic to plants.

公开(公告)号：EP1662877A1

公开(公告)日：2006-06-07

申请号：EP04765059.3

申请日：2004-09-10

申请人： BASF Aktiengesellschaft

发明人： BAUMANN, Ernst ,  GROTE, Thomas ,  SCHIEWECK, Frank ,  VON DEYN, Wolfgang ,  GÖTZ, Norbert ,  HOFMANN, Michael ,  KORDES, Markus ,  PUHL, Michael ,  RACK, Michael ,  SCHMIDT, Thomas ,  BUCCI, Toni ,  COTTER, Henry, Van, Tuyl ,  CULBERTSON, Deborah, L. ,  OLOUMI-SADEGHI, Hassan

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The present invention relates to a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one 6-halogeno [1,2,4]-triazolo[1,5-a]-pyrimidine of the general formula (I), wherein X, R1, R2 , R3 and R4 are as defined in claim 1 and/or the agriculturally useful salts thereof.

公开(公告)号：EP1504009A1

公开(公告)日：2005-02-09

申请号：EP03747437.6

申请日：2003-04-30

申请人： BASF AKTIENGESELLSCHAFT

发明人： TORMO I BLASCO, Jordi ,  BLETTNER, Carsten ,  MÜLLER, Bernd ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  GYPSER, Andreas ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried ,  LORENZ, Gisela ,  STIERL, Reinhard

IPC分类号： C07D487/04 ,  A01N43/90 ,  C07C69/612 ,  C07C69/65 ,  C07C69/738

CPC分类号： C07D487/04 ,  A01N43/90 ,  C07C69/65

摘要： Disclosed are a method for producing fungicidal triazolopyrimidine compounds, agents containing said compounds, and the use thereof for controlling harmful fungi. Also disclosed are triazolopyrimidines of formula (I), in which the substituents have the following meaning: L1 represents alkyl; L2 represents halogen; L3 represents hydrogen or halogen; X represents halogen, cyano, alkyl, alkoxy, or haloalkoxy; R1, R2 represent hydrogen, alkyl, haloalkyl, cycloalkyl, alkenyl, alkadienyl, alkinyl, or cycloalkinyl, phenyl, naphthyl, or a five-unit to ten-unit saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group O, N, or S. R1 and R2 can also form a five-unit or six-unit ring along with the nitrogen atom to which they are linked. Said ring can be interrupted and/or substituted by an atom from the group O, N, and S while R1 and/or R2 can be substituted according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing said compounds, and the use thereof for controlling harmful fungi.