N- [ (PYRIDIN- 2 -YL) METHOXY]HETEROCYCLYL CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS FUNGICIDES
    5.
    发明公开
    N- [ (PYRIDIN- 2 -YL) METHOXY]HETEROCYCLYL CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS FUNGICIDES 审中-公开
    N - [(吡啶-2-基)甲氧基]HETEROCYCLYLCARBONSÄUREAMIDDERIVATE及相关化合物作为杀真菌剂

    公开(公告)号:EP2041092A1

    公开(公告)日:2009-04-01

    申请号:EP07787095.4

    申请日:2007-07-05

    IPC分类号: C07D213/61

    摘要: A compound of general formula (I): in which: - n is 1,2,3 or 4; - X is a halogen atom, a nitro group, a cyano group, a hydroxy group, an amino group, a sulfanyl group, a pentafluoro- λ6-sulfanyl group, a formyl group, a formyloxy group, a formylamino group, a carboxy group, a carbamoyl group, a N-hydroxycarbamoyl group, a carbamate group, a (hydroxyimino)-C1C6-alkyl group, a C1-C-aIkyI, a C2-C8-alkenyl, a C2-C8-alkynyl, a tri(C1-C8-alkyl) silyl, a C1 -C8-alkylamino, a di-C1-C8-alkylamino, a C1-C8-alkoxy, a C1-C8-haloalkyl group, a C1-C8-halogenoalkoxy having 1 to 5 halogen atoms, - A is an oxygen atom, a NR3 group, a sulphur atom, a sulphinyl group, a sulphonyl group or a SiR4R5 group; - R1 and R2 are chosen independently of each other as being a hydrogen atom, a halogen atom, a cyano group, a hydroxy group, an amino group, a sulfanyl group, a formyl group, a formyloxy group, a formylamino group, a carboxy group, a carbamoyl group, a N-hydroxycarbamoyl group, a carbamate group, a (hydroxyimino)-C1-C6-alkyl group, a C1-C6-alkyl, a C2-C6-alkenyl, a C2-C6--alkynyl, - R3 is a hydrogen atom, a C1-C6--alkyl, or a C3-C7-CycloaIkyI; - R4 and R5 are chosen independently of each other as being a hydrogen atom, a cyano group, a hydroxy group, a formyl group, a C1-C6-aIkyl, a C2-C6-alkenyl, - Het represents a 5-, 6- or 7-membered non-fused heterocycle with one, two or three heteroatoms which ma be the same or different, Het being linked by a carbon atom and Het being optionally substituted by one or further substituents A process for preparing this compound. A fungicidal composition comprising a compound of general formula (I)- A method for treating plants by applying a compound of general formula (I) or a composition comprising it.

    METHOD FOR IDENTIFICATION OF NOVEL FUNGICIDES
    6.
    发明公开
    METHOD FOR IDENTIFICATION OF NOVEL FUNGICIDES 审中-公开
    方法识别新型杀菌剂

    公开(公告)号:EP1893771A1

    公开(公告)日:2008-03-05

    申请号:EP06763587.0

    申请日:2006-06-08

    IPC分类号: C12Q1/18

    CPC分类号: G01N33/56961

    摘要: The present invention deals with a method for identifying fungicidal compounds comprising the steps of : contacting fungal cells with said compound, contacting said fungal cells with an antibody raised against spectrin protein, and observing the distribution of spectrin-like proteins relative to a control, wherein the redistribution of the spectrin-like protein from a inner face of cell membrane to a cytosolic location identifies a fungicide candidate.