公开(公告)号：EP1970372B1

公开(公告)日：2010-11-03

申请号：EP06843969.4

申请日：2006-11-17

申请人： EPhaG AS

发明人： SURKOV, Kirill Gennadievich

IPC分类号： C07D219/06 ,  C07H5/06 ,  A61K31/435 ,  A61P31/12 ,  A61P33/00 ,  A61P37/02

CPC分类号： C07D219/06

摘要： The invention relates to 1-alkylamino-1-desoxy-polyols and 9-oxoacridine-10-acetic acid salts of general formula (I), wherein A is (II), in which R is selected from an ethyl, propyl and butyl group, to medicinal preparations containing an active agent embodied in the form of one or several salts of formula (1) according to item 1 and/or the mixture of said salt of formula (I) or the 9-oxoacridine-10-acetic acid of formula (III) with one or several 1-alkylamino-1-desoxy-polyols of general formula (II), wherein R is selected from the ethyl, propyl and butyl group.

摘要翻译： 本发明涉及通式（I）的1-烷基氨基-1-脱氧 - 多元醇和9-氧代吖啶-10-乙酸盐，其中A是（II），其中R选自乙基，丙基和丁基 涉及含有以一种或多种根据第1项的式（1）的盐形式包含的活性剂和/或所述式（I）的盐或式（I）的盐的混合物的9-氧代吖啶-10-乙酸 （III）与一种或多种通式（II）的1-烷基氨基-1-脱氧 - 多元醇反应，其中R选自乙基，丙基和丁基。

公开(公告)号：EP1970372A2

公开(公告)日：2008-09-17

申请号：EP06843969.4

申请日：2006-11-17

申请人： EPhaG AS

发明人： SURKOV, Kirill Gennadievich

IPC分类号： C07D219/06 ,  C07H5/06 ,  A61K31/435 ,  A61P31/12 ,  A61P33/00 ,  A61P37/02

CPC分类号： C07D219/06

摘要： The invention relates to salts of 1-alkylamino-1-deoxypolyols and 9-oxoacridine-10-acetic acid of the general formula (I):

wherein A + is (II)

wherein R is selected from the group consisting of ethyl, propyl, butyl,
medicinal preparations comprising as an active ingredient salts of formula (I) and/or a mixture of said salt of formula (I) or 9-oxoacridine-10-acetic acid of the formula:

and one or more 1-alkylamino-1-deoxypolyols of the general formula (II):

wherein:
R is selected from the group consisting of ethyl, propyl, butyl.

摘要翻译： 本发明涉及通式（I）的1-烷基氨基-1-脱氧多羟基化合物和9-氧代吖啶-10-乙酸的盐：其中A +是（II）其中R选自乙基，丙基，丁基 包含作为活性成分的式（I）的盐和/或所述式（I）的盐或下式的9-氧代吖啶-10-乙酸与一种或多种1-烷基氨基-1- 通式（II）的脱氧多羟基化合物：其中：R选自乙基，丙基，丁基。