公开(公告)号：EP0861242A1

公开(公告)日：1998-09-02

申请号：EP96933541.0

申请日：1996-10-11

申请人： AgrEvo UK Limited

发明人： O'MAHONY, Mary Josephine, Chesterford Park ,  WEST, Peter John, Chesterford Park ,  MACRITCHIE, Jacqueline Anne, Chesterford Park ,  MILLWARD, Peter

IPC分类号： C07H17 ,  A01N43 ,  A01N55 ,  C07D311 ,  C07D405 ,  C07D407 ,  C07D413 ,  C07D417

CPC分类号： C07D311/18 ,  A01N43/16 ,  C07D311/22 ,  C07D311/54 ,  C07D311/56

摘要： Compounds of forumla (I) where one of Z and Y is CO and the other is C-W-R2 and the dotted line indicates a double bond is present where necessary to meet valency requirements, W is O, S(O)¿n?, N(R?3), N(R3)N(R4), N(R3¿)O or ON(R3); R1 is hydrogen, or an optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, phenyl or heterocyclyl group; R?2, R3 and R4¿, which may be the same or different, are as defined above for R1, or are acyl, or R?2 and R3 or R2 and R4 or R3 and R4¿ together with the nitrogen or oxygen to which they are attached form an optionally substituted ring which may contain other hetero atoms; each X, which may be the same as or different from any other X, is halogen, CN, NO¿2?, SF5, B(OH)2, trialkylsilyl or a group E, OE or S(O)nE where E is a group as defined hereinbefore for R?2¿ or is optionally substituted amino; or two adjacent groups X together with the atoms to which they are attached form an optionally substituted carbocyclic or heterocyclic ring; n is 0, 1 or 2; and p is 0 to 4 have fungicidal activity. Many of the compounds are novel.

摘要翻译： 其中Z和Y之一是CO且另一个是CW-R2且虚线表示双键的论坛（I）化合物在必要时存在以满足化合价要求，W是O，S（O）n'， N（R 3），N（R 3）N（R 4），N（R 3'）O或ON（R 3）。 R 1是氢或任选取代的烷基，烯基，炔基，环烷基，苯基或杂环基; R 2，R 3和R 4可以相同或不同，如上面对R 1定义的，或者是酰基，或R 2和R 3或R 2和R 4或R 3和R 4'与氮或氧一起形成 它们连接形成可含有其它杂原子的任选取代的环; 每个X可与任何其它X相同或不同，为卤素，CN，NO2，SF5，B（OH）2，三烷基甲硅烷基或基团E，OE或S（O）nE，其中E为 如上所定义的基团，R 2'或是任选取代的氨基; 或两个相邻基团X与它们所连接的原子一起形成任选取代的碳环或杂环; n是0,1或2; 并且p是0至4具有杀真菌活性。 许多化合物都是新颖的。