公开(公告)号：EP2105442A1

公开(公告)日：2009-09-30

申请号：EP07850951.0

申请日：2007-12-20

申请人： Astellas Pharma Inc. ,  Kotobuki Pharmaceutical Co., Ltd.

发明人： KOMENOI, Kousuke ,  NAKAMURA, Atsushi ,  KASAI, Makoto ,  IMAMURA, Masakazu ,  SHIRAKI, Ryota ,  NAKANISHI, Keita

IPC分类号： C07D409/10 ,  A61K31/381 ,  A61P3/10 ,  C07D333/54

CPC分类号： C07D409/10 ,  C07D333/54

摘要： The present invention provides a method for producing a C-glycoside derivative, which can produce the C-glycoside derivative at a high yield and at a low cost, which conforms to environmental protection, and which is applicable industrially. The C-glycoside derivative is useful for treating and preventing diabetes such as insulin-dependent diabetes (type 1 diabetes), non-insulin-dependent diabetes (type 2 diabetes) and the like and various diabetes-related diseases including insulin-resistant diseases and obesity.

摘要翻译： 本发明提供一种可以以高产率和低成本生产符合环境保护并且在工业上可应用的C-糖苷衍生物的方法。 C-糖苷衍生物可用于治疗和预防糖尿病如胰岛素依赖性糖尿病（1型糖尿病），非胰岛素依赖型糖尿病（2型糖尿病）等，以及各种糖尿病相关疾病，包括胰岛素抵抗性疾病和 肥胖。