公开(公告)号：EP0631575B1

公开(公告)日：2001-10-04

申请号：EP93906495.2

申请日：1993-03-10

申请人： Aventis CropScience GmbH

发明人： SCHAPER, Wolfgang ,  FREUSS, Rainer ,  SALBECK, Gerhard ,  BRAUN, Peter ,  KNAUF, Werner ,  SACHSE, Burkhard ,  WALTERSDORFER, Anna ,  KERN, Manfred ,  LÜMMEN, Peter, Dr. ,  BONIN, Werner

IPC分类号： C07D239/46 ,  C07D239/42 ,  C07D239/52 ,  C07D239/34 ,  C07D239/94 ,  C07D239/88 ,  C07D401/12 ,  C07D495/04

CPC分类号： C07D239/34 ,  A01N43/54 ,  A01N43/90 ,  C07D239/42 ,  C07D239/47 ,  C07D239/52 ,  C07D239/88 ,  C07D239/94 ,  C07D401/12 ,  C07D405/12 ,  C07D495/04

公开(公告)号：EP1100785A1

公开(公告)日：2001-05-23

申请号：EP99941447.7

申请日：1999-07-20

申请人： Aventis CropScience GmbH

发明人： MÄRKL, Martin ,  SCHAPER, Wolfgang ,  ORT, Oswald ,  JAKOBI, Harald ,  BRAUN, Ralf ,  KRAUTSTRUNK, Gerhard ,  SANFT, Ulrich ,  BONIN, Werner ,  STARK, Herbert ,  PASENOK, Sergej ,  CABRERA, Ivan

IPC分类号： C07D239/42 ,  C07D239/46 ,  A01N43/54

CPC分类号： C07D239/42 ,  A01N43/54 ,  C07D239/47

摘要： Compounds of formula (I) where R1 is hydrogen, chlorine, fluorine or methyl, R?2 and R3¿, which may be the same or different from each other, are hydrogen, halogen, cyano, (C¿1?-C4)-alkyl, vinyl, ethynyl, (C1-C4)-alkoxy, (C1-C4)-alkoxy-(C1-C4)-alkyl, fluorovinyl or fluoroethyl, or R?2 and R3¿ together with the linking carbon atoms form a benzo ring, and R4 is (C¿2?-C4)-alkyl, (C2-C4)-alkenyl or (C3-C4)-alkinyl, each of which is substituted by at least two fluorine atoms and optionally substituted by C1-4-alkoxy, cyanomethoxy, (C3-C4)-alkenyloxy or (C3-C4)-alkinyloxy, are useful as pesticides, especially against insects, acarids and fungi. The invention includes a novel process for fluorinating certain pyrimidines.

摘要翻译： 其中R 1为氢，氯，氟或甲基，R 2和R 3可相同或不同的式（Ⅰ）化合物是氢，卤素，氰基，（C 1 -C 4） （C 1 -C 4） - 烷氧基，（C 1 -C 4） - 烷氧基 - （C 1 -C 4） - 烷基，氟乙烯基或氟乙基，或者R 2和R 3与连接的碳原子一起形成 苯并环，并且R 4是（C 2 -C 4） - 烷基，（C 2 -C 4） - 烯基或（C 3 -C 4） - 炔基，其各自被至少两个氟原子取代并且任选被C 1 -C 4 - （C 3 -C 4） - 链烯氧基或（C 3 -C 4） - 炔氧基，可用作杀虫剂，特别是对昆虫，螨和真菌。 本发明包括氟化某些嘧啶的新方法。

公开(公告)号：EP1068197A1

公开(公告)日：2001-01-17

申请号：EP99916871.9

申请日：1999-03-23

申请人： Aventis CropScience GmbH

发明人： SCHAPER, Wolfgang ,  BRAUN, Ralf ,  JAKOBI, Harald ,  KRAUTSTRUNK, Gerhard ,  MÄRKL, Martin ,  ORT, Oswald ,  KERN, Manfred ,  SANFT, Ulrich ,  BONIN, Werner

IPC分类号： C07D401/12 ,  A01N43/54 ,  A01N43/40 ,  C07D409/14 ,  C07D401/14

CPC分类号： C07D401/12 ,  A01N47/16 ,  A01N47/38 ,  C07D401/14 ,  C07D405/14 ,  C07D409/14

摘要： The invention relates to substituted piperidines of formula (I), wherein R1 represents H, halogen, alkyl, alkyl halide or cycloalkyl; R?2 and R3¿ have the meaning given in the description; A represents CH or N; X represents NH, O or S(O)¿q?, q being equal to 0, 1 or 2; Y and Z represent O, S or optionally substituted imino; m and n are equal to 1, 2, 3, 4, or 5; R?4 and R4'¿ represent H, alkyl, alkyl halide, halogen or alkoxy; R5 represents one or more of the following optionally substituted groups: alkyl, alkenyl, alkynyl, aryl or heterocyclyl, one or more C-units which can be substituted with CO or heteroatom-units. The invention also relates to a method for preparing said compounds, agents containing them and their use as pesticides and fungicides.