公开(公告)号：EP0982992B1

公开(公告)日：2002-09-25

申请号：EP98919374.3

申请日：1998-05-01

申请人： Aventis CropScience UK Limited

发明人： ATHERALL, John, Frederick ,  HOUGH, Thomas, Lawley ,  LINDELL, Stephen, David ,  O'MAHONY, Mary, Josephine ,  SAVILLE-STONES, Elizabeth Anne ,  PARSONS, John Henry

IPC分类号： A01N43/90 ,  C07D495/04

CPC分类号： C07D495/04 ,  A01N43/90

摘要： The invention provides the use in combating fungi of compounds of general formula (I) wherein R1 is hydrogen, hydroxy, acyl, acyloxy, optionally substituted amino, Ra, Ra3Si, RaS or RaO, where Ra is optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted cycloalkyl, optionally substituted cycloalkenyl, optionally substituted aryl or optionally substituted heterocyclyl; R2 has the same meaning as Ra or can be hydrogen; Z is oxygen or sulfur; M is a thiophene ring; and R?3 and R4¿, which may be the same or different, have the same meaning as Ra or can be optionally substituted amino, hydrogen, halogen, cyano, nitro or a group ORc or S(O)¿mR?c, where Rc has the same meaning as Ra or is hydrogen or acyl and m is 0, 1 or 2; or R?3 and R4¿ together with the atoms to which they are attached form an optionally substituted carbocyclic or heterocyclic ring; together with tautomers of compounds where R1 is hydrogen.

公开(公告)号：EP0861242B1

公开(公告)日：2001-05-30

申请号：EP96933541.3

申请日：1996-10-11

申请人： Aventis CropScience UK Limited

发明人： O'MAHONY, Mary Josephine, Chesterford Park ,  WEST, Peter John, Chesterford Park ,  MACRITCHIE, Jacqueline Anne, Chesterford Park ,  LINDELL, Stephen, David ,  MILLWARD, Peter

IPC分类号： C07D311/22 ,  C07D311/54 ,  C07D311/56 ,  C07D311/18 ,  A01N43/16

CPC分类号： C07D311/18 ,  A01N43/16 ,  C07D311/22 ,  C07D311/54 ,  C07D311/56

摘要： Compounds of forumla (I) where one of Z and Y is CO and the other is C-W-R2 and the dotted line indicates a double bond is present where necessary to meet valency requirements, W is O, S(O)¿n?, N(R?3), N(R3)N(R4), N(R3¿)O or ON(R3); R1 is hydrogen, or an optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, phenyl or heterocyclyl group; R?2, R3 and R4¿, which may be the same or different, are as defined above for R1, or are acyl, or R?2 and R3 or R2 and R4 or R3 and R4¿ together with the nitrogen or oxygen to which they are attached form an optionally substituted ring which may contain other hetero atoms; each X, which may be the same as or different from any other X, is halogen, CN, NO¿2?, SF5, B(OH)2, trialkylsilyl or a group E, OE or S(O)nE where E is a group as defined hereinbefore for R?2¿ or is optionally substituted amino; or two adjacent groups X together with the atoms to which they are attached form an optionally substituted carbocyclic or heterocyclic ring; n is 0, 1 or 2; and p is 0 to 4 have fungicidal activity. Many of the compounds are novel.