PYRIDYLESSIGSÄUREDERIVATE, VERFAHREN UND ZWISCHENPRODUKTE ZU IHRER HERSTELLUNG UND SIE ENTHALTENDE MITTEL
    5.
    发明公开
    PYRIDYLESSIGSÄUREDERIVATE, VERFAHREN UND ZWISCHENPRODUKTE ZU IHRER HERSTELLUNG UND SIE ENTHALTENDE MITTEL 失效
    PYRIDYLESSIGSÄUREDERIVATE,工艺以及它们和代理人含相同的中间产品

    公开(公告)号:EP0876344A1

    公开(公告)日:1998-11-11

    申请号:EP96937262.0

    申请日:1996-10-28

    IPC分类号: C07D213 A01N43

    CPC分类号: C07D213/54

    摘要: The invention concerns pyridylacetic acid derivatives of formula (I), in which the substituents and the index have the following meanings: X - NOCH3, CHOCH3, CHCH3 and CHCH2CH3; Y - oxygen or NR', R' representing hydrogen or alkyl; R - cyano, nitro, trifluoromethyl, halogen, alkyl and alkoxy; m is 0, 1 or 2; R1 is hydrogen and alkyl; R2 - hydrogen, cyano, nitro, hydroxy, amino, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkyl thio, alkylamino or dialkylamino; R3 - hydrogen, cyano, nitro, hydroxy, amino, halogen; or optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenyl, alkenyloxy, alkenylthio, alkenylamino, N-alkenyl-N-alkylamino, alkinyl, alkinyloxy, alkinylthio, alkinylamino, N-alkinyl-N-alkylamino, cycloalkyl, cycloalkyloxy, cycloalkylthio, cycloalkylamino, N-cycloalkyl-N-alkylamino, cycloalkenyl, cycloalkenyloxy, cycloalkenylthio, cycloalkenylamino, N-cycloalkenyl-N-alkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio, heterocyclylamino, N-heterocyclyl-N-alkylamino,aryl, aryloxy, arylthio,arylamino, N-aryl-N-alkylamino, hetaryl, hetaryloxy, hetarylthio, hetarylamino, and N-hetaryl-N-alkylamino; R4 - hydrogen, optionally substituted alkyl, alkenyl, alkinyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, alkylsulphonyl, cycloalkyl, aryl, arylcarbonyl, arylsulphonyl, hetaryl, hetarylcarbonyl, or hetarylsulphonyl. Also disclosed are the salts of the above derivatives,and methods and intermediate products for producing them and agents containing them.